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2-(2-hydroxyethyl)-9-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]ethan-1-one
2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}-5-methylphenol
4-chloro-1,5-dimethyl-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-1H-pyrazole-3-carboxamide
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-2-methyl-1,3-thiazole-4-carboxamide
1-cyclohexyl-5-(1,4-dioxan-2-yl)-3-[(2-methoxyphenyl)methyl]-1H-1,2,4-triazole
5-(2-methyl-1,4-oxazepane-4-carbonyl)-2-(pyridin-3-yl)pyrimidin-4-ol
1-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-1-methyl-3-[4-methyl-3-(propan-2-yl)phenyl]urea
(2S,4S)-4-amino-1-(1-benzoxepine-4-carbonyl)-N-ethylpyrrolidine-2-carboxamide
5-{[(1S,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
4-{3-[2-(3-fluorophenyl)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
2-{1-[(3-methoxyphenyl)methyl]-4-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
N-[2-(pyridin-3-ylformamido)ethyl]cyclohex-3-ene-1-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carboxamide
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-1-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}propan-1-one
N-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)ethyl]-6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-methoxy-4-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
5-(1H-imidazol-1-ylmethyl)-3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazole
5-(3,4-dimethylphenoxymethyl)-N-ethyl-N-(pyridin-4-ylmethyl)-1,2-oxazole-3-carboxamide
1-({[1-(3-fluoro-4-hydroxyphenyl)ethyl]carbamoyl}methyl)piperidine-4-carboxamide
N-[(5-methylpyrazin-2-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
(1R,2S,4R)-N-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(3R,4S)-1-(oxan-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-2-(4H-1,2,4-triazol-4-yl)acetamide
3-methyl-1-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]-3-phenylpiperidine
5-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine-2-carbonitrile
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-1-[4-(thiophene-2-carbonyl)piperazin-1-yl]propan-1-one
5-[(3-fluorophenyl)methyl]-3-(2-methoxyethyl)-5-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-2-(pyridin-4-yl)quinoline-4-carboxamide
3-[1-(cyclohexylmethyl)-1H-pyrazol-5-yl]-1-ethyl-1-(oxan-4-ylmethyl)urea
1-{4-[2-(3,4-dimethoxyphenyl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}pent-4-en-1-one
5-(azepane-1-carbonyl)-1-(butan-2-yl)-4-oxo-N-{[4-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
4-(2-oxo-2-{4-[(2-oxopyrrolidin-1-yl)methyl]piperidin-1-yl}ethyl)-4-azatricyclo[4.3.1.13,8]undecan-5-one
1-{[2-(4-ethoxyphenoxy)phenyl]methyl}-4-methylpiperazine
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-5-(2-fluorophenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
1-{3-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-3-oxopropyl}azepan-2-one
N-(thiolan-3-yl)-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
8-[2-(azepan-1-yl)acetyl]-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2R)-2-({4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)-2-phenylethan-1-ol
1,9-dimethyl-4-[4-(4-methylphenyl)-4-oxobutyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
3-{3-benzyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-5-(propan-2-yl)-1,2-oxazole
1-(2-fluorophenyl)-4-(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)piperazine
1-[2-(dimethylamino)-4-({[3-(methylsulfanyl)phenyl]methyl}amino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
2-[2-oxo-4-(pyrazine-2-carbonyl)piperazin-1-yl]benzonitrile
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(1H-indol-1-yl)ethan-1-one
3-{[(cyclopropylcarbamoyl)methyl]sulfamoyl}-N-methyl-N-[2-(methylsulfanyl)ethyl]benzamide
2-{4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
methyl 1-[(3S,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide