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3-methoxy-2-({3-[(4-methoxyphenyl)amino]piperidin-1-yl}methyl)phenol
ethyl 4-[(4-chlorophenyl)methyl]-1-{[4-(2-hydroxyethoxy)phenyl]methyl}piperidine-4-carboxylate
2-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-{[(2S,4R)-4-cyclobutaneamido-2-(ethylcarbamoyl)pyrrolidin-1-yl]methyl}benzoic acid
(3S,4R)-1-(5-fluoro-3-methyl-1H-indole-2-carbonyl)-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
5-cyclopropanecarbonyl-1'-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-3-(4-methylphenyl)propanamide
3-{3-[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]phenyl}-5-methyl-4H-1,2,4-triazole
4-[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridine-6-carbonyl]-7-fluoro-1,2-dihydroquinolin-2-one
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[2-(pyrazin-2-yl)ethyl]piperidine-4-carboxamide
1-[3-(1-benzofuran-2-yl)-1-methyl-1H-1,2,4-triazol-5-yl]piperidine
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}propanamide
1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-(2-phenylethyl)piperidine
methyl (2S,4S,5R)-5-(4-chlorophenyl)-4-[(cyclopropylmethyl)carbamoyl]-1,2-dimethylpyrrolidine-2-carboxylate
2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-2-phenyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}acetamide
1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-4-phenylpyrrolidin-2-one
1-phenyl-N-[(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)methyl]methanesulfonamide
N-methyl-2-(1H-pyrazol-1-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
1-[1-(2-ethylbutyl)piperidin-4-yl]-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
(1R,2S,6R,7S)-4-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-azatricyclo[5.2.2.02,6]undecane
(1S,4S)-2-[2-(methylsulfanyl)phenyl]-5-[2-(trifluoromethyl)benzoyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
(2S)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-acetamido-4-(methylsulfanyl)butanamide
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylacetamide
1'-[4-(1H-1,2,4-triazol-3-yl)benzoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-(2-methyl-1H-imidazol-1-yl)-N-[4-(3-methylphenyl)-1-phenyl-1H-pyrazol-5-yl]acetamide
4-hydroxy-N,2-dimethyl-N-{[3-(methylsulfanyl)phenyl]methyl}pyrimidine-5-carboxamide
(2S,4S)-4-amino-1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}(methyl)[3-(1H-pyrazol-1-yl)propyl]amine
3-phenyl-7-{1H-pyrrolo[2,3-b]pyridin-6-yl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
1-{4-[(pentan-3-yl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2,5-dihydro-1H-pyrrole-2-carboxamide
(5S)-5-{[benzyl({[6,7-dimethoxy-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl})amino]methyl}pyrrolidin-2-one
N-benzyl-N-ethyl-5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2-oxazole-3-carboxamide
4-(1,3-benzothiazol-2-ylmethyl)-9-methoxy-7-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})[(1-methyl-1H-imidazol-2-yl)methyl]amine
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
5,6-dimethyl-2-oxo-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,2-dihydropyridine-3-carboxamide
1-propyl-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidin-4-amine
1-[(3,5-dimethylphenyl)methyl]-4-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]piperazin-2-one
3-(2-fluorophenyl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
1-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-hydroxy-4-methylpentan-1-one
N,N-diethyl-1-{[1-(2-methylpropanoyl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
3-[(3R,4S)-4-(dimethylamino)-1-[(2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)sulfonyl]piperidin-3-yl]propanoic acid
2-(3-fluorophenyl)-5-(1,2,3-thiadiazol-4-yl)-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)-5-(propan-2-yl)-1,3-oxazole-4-carboxamide
3-[(3R,4S)-3-[(6-cyclopropylpyrimidin-4-yl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]propanamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)oxane-4-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
(4aR,7aS)-1-ethyl-4-{[3-(5-methylfuran-2-yl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(2-ethylmorpholin-4-yl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene