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4-{1-[5-(1H-imidazol-2-yl)thiophene-2-carbonyl]piperidin-4-yl}thiomorpholine
1-cyclobutanecarbonyl-N-{[4-(methylsulfanyl)phenyl]methyl}piperidine-4-carboxamide
2-[(3-cyclopentyl-1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-5,6-dimethyl-2,3-dihydropyridazin-3-one
2-(2,3-difluoro-6-methoxybenzoyl)-octahydropyrrolo[1,2-a]piperazine
1-(2,5-dimethoxybenzoyl)-N-(4-fluorophenyl)piperidin-3-amine
6-(2-chlorophenyl)-N-methyl-N-[(3-methylpyridin-4-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-1-(2-methoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
1-[1-(3,5-dimethylfuran-2-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[(2E)-3-phenylprop-2-enoyl]piperidin-3-yl]propanoic acid
N-[(3S,4R)-4-(4-methoxyphenyl)-1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)pyrrolidin-3-yl]acetamide
methyl 3-[(3S,4R)-4-(dimethylamino)-1-[(3-hydroxyphenyl)methyl]piperidin-3-yl]propanoate
3-(3,5-dimethoxyphenyl)-6-methoxypyridazine
2-(2,2-dimethylpropanamido)-5-methyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]thiophene-3-carboxamide
4-({[1-(ethylcarbamoyl)piperidin-4-yl]amino}methyl)-2,6-dimethylphenyl acetate
N,2-dimethyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-6-(piperidin-3-yl)pyrimidin-4-amine
7-(2,2-dimethylpropyl)-2-(1,3-thiazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-[(4-chlorophenyl)methyl]-8-[(2S)-2-hydroxypropanoyl]-2,8-diazaspiro[4.5]decan-3-one
3-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
3-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1-[4-(propylsulfamoyl)phenyl]urea
12-[4-(2-methoxyethyl)piperazine-1-carbonyl]-15-methyl-9-(pyridin-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaen-13-one
5-cyclopropyl-N-[2-(dimethylamino)ethyl]-N-methyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-[(3R,4R)-3-[(4-ethylpiperazin-1-yl)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]pyridine-4-carboxamide
(2S,4S)-4-amino-N-ethyl-1-[5-(propan-2-yl)pyrimidin-4-yl]pyrrolidine-2-carboxamide
3-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-1-methyl-1H-indazole
1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-3-[3-(propan-2-yloxy)benzoyl]piperidine
3-methyl-1-({1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}methyl)-1H-pyrazol-5-amine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylcyclopropanesulfonamide
2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]-1-[7-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
N,1-dimethyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidine-2-carboxamide
4-methyl-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]pyridine-3-carboxamide
2,3-dimethyl-6-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-2-(1H-imidazol-1-yl)-N-(pyridin-4-ylmethyl)acetamide
3-{1-[2-(dimethyl-1H-1,2,4-triazol-1-yl)acetyl]piperidin-3-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
methyl({[2-(propan-2-yl)pyrimidin-4-yl]methyl}){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
methyl 3-(2H-1,3-benzodioxol-4-ylmethyl)-7-oxo-9-(thiophen-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(3,6-dimethylpyrazin-2-yl)-4-[3-(furan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
(3S,4R)-3-ethyl-4-methyl-1-[2-(morpholin-4-yl)pyridine-3-carbonyl]piperidin-4-ol
(3S,4R)-1-(2-carboxyethyl)-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
({6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}methyl)[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]methylamine
(2S,4S)-4-cyclopentaneamido-N,N-diethyl-1-(thiophen-2-ylmethyl)pyrrolidine-2-carboxamide
(1S,2S,9S)-N-[3-(dimethylamino)phenyl]-6-oxo-7,11-diazatricyclo[7.3.1.02,7]tridecane-11-carboxamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]acetamide
2-(1-{[1-(6-methylhept-5-en-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-(pyridin-4-ylmethyl)-4-[1-(pyridine-2-carbonyl)piperidin-4-yl]-1,4-diazepane
2-[(2-methoxyethyl)(methyl)amino]-2-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]acetic acid
(3R,4S)-4-(3-methoxyphenyl)-1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)pyrrolidin-3-amine
1-[2-(dimethylamino)-6-(1H-pyrazole-3-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl]piperidin-4-ol
5-tert-butyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]-1,3,4-oxadiazol-2-amine