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5-cyclohexaneamido-N-[(3,5-difluorophenyl)methyl]-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carboxamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-1-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethan-1-one
N-[1-(2-chlorophenyl)ethyl]-5-acetamido-1-(2-methoxyethyl)-2-(pyridin-2-yl)-1H-1,3-benzodiazole-7-carboxamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(1-methylpiperidin-2-yl)propanamide
N-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
9-methoxy-N-methyl-7-oxo-3-(2,2,3,3-tetramethylcyclopropanecarbonyl)-N-(1,3-thiazol-4-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
6-methyl-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}-1,3-benzothiazole
2-[(3-methoxyphenyl)amino]-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propylbutanamide
methyl({[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}){[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}amine
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-propoxybenzamide
methyl 4-{[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
3-methyl-6-{5-[1-(1H-1,2,4-triazol-1-yl)ethyl]-1,2,4-oxadiazol-3-yl}pyridazine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-(4-methylpiperazin-1-yl)pentanamide
4-(5-phenyl-1,2-oxazole-3-carbonyl)-7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
(7S,9aR)-7-[(2S)-butan-2-yl]-N-cyclohexyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
4-(1-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
3-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]-1-{2-[2-(trifluoromethoxy)phenyl]ethyl}urea
2-(4-cyclopentyl-1,4-diazepan-1-yl)-2-(5-fluoro-2-methoxyphenyl)acetic acid
5-(3-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-3-oxopropyl)-5-[(4-phenylphenyl)methyl]pyrrolidin-2-one
ethyl[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
4-ethyl-N,N-dimethyl-6-[3-(1H-pyrazol-5-yl)piperidin-1-yl]pyrimidin-2-amine
propyl 2-cyclopropyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxylate
N4-[2-(dimethylamino)-1-phenylethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-phenyl-N-{1-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
5-(4-{[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)-1H-indole
5-(5-methyl-4-phenylthiophene-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(2-methylphenyl)acetamide
3-[(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)amino]butan-1-ol
1-(piperazin-1-yl)-3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)propan-2-ol
1-(3-fluorophenyl)-6,6-dimethyl-N-(thian-4-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-methyl-6-(propan-2-yl)-N-[3-(4H-1,2,4-triazol-4-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(3R,4S)-1-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
7-[2-(azepan-1-yl)acetyl]-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(4-methoxypyridin-2-yl)methyl]-2-methylthieno[3,2-d]pyrimidin-4-amine
1-methyl-4-(1-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}ethyl)piperazine
1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}urea
2-{4-[4-(2-methoxyphenoxy)piperidin-1-yl]piperidin-1-yl}-4,6,7-trimethylquinazoline
(2S,4S)-4-[(naphthalen-1-ylmethyl)amino]-N-(propan-2-yl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-[2-(3,4-dimethylphenyl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N,N-bis(2-hydroxyethyl)-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-(thiolan-3-yl)propanamide
3-(1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)pyridine
(1S,5R)-3-[2-(4-fluorophenyl)acetyl]-3,9-diazabicyclo[3.3.2]decan-10-one
N-methyl-3-[(2-methylprop-2-en-1-yl)oxy]-N-[(5-propyl-1H-pyrazol-3-yl)methyl]benzamide
1-(3-chlorophenyl)-4-(2,3-difluorobenzoyl)piperazin-2-one
1-(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)piperazine
2-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
3-{[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}pyridin-2-ol
2-amino-6-{4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperazin-1-yl}-3,4-dihydropyrimidin-4-one