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N-cyclopentyl-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
2-[7-(hydroxymethyl)-9-(1H-imidazol-2-ylmethyl)-3,9-diazaspiro[5.5]undecan-3-yl]acetic acid
5-(4-methyl-1H-imidazol-5-yl)-1-(oxan-4-ylmethyl)-4-phenyl-1H-imidazole
3-(3-methoxyphenyl)-5-(3-methylfuran-2-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
(1R,3S)-3-(2-hydroxyethoxy)-7-(1,2-thiazole-5-carbonyl)-7-azaspiro[3.5]nonan-1-ol
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperidine
5-(2-butoxyphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
diethyl({[3-(4-methyl-1,4-diazepane-1-carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]methyl})amine
methyl (2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxylate
8-methyl-3-{2-[methyl(2-phenylethyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]-5-(trifluoromethyl)pyridine
N3-benzyl-N5-cycloheptyl-N3-(2-hydroxyethyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-2-(1-ethylpiperidin-4-yl)acetamide
N5-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N3,N3-dimethyl-1,2,4-thiadiazole-3,5-diamine
(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
4-[1-(cyclopentylmethyl)pyrrolidin-3-yl]-2-(2,6-dimethoxyphenyl)pyridine
3-({1-[2-(methylamino)-1,3-thiazole-4-carbonyl]piperidin-4-yl}methyl)benzoic acid
1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-N-{[2-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
2-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]pyridine-3-carbonitrile
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(3-hydroxy-1,2-oxazol-5-yl)-N-methylpropanamide
2-[3-(1-methyl-1H-pyrazol-3-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]propanoic acid
1-(3-methanesulfonamidophenyl)-3-(3-methoxypropyl)urea
7-[(4-ethylphenyl)methyl]-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
2-{[2-(pyridin-4-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-tert-butyl-3-[(3,4-dimethoxyphenyl)methyl]-5-(5-methyl-1,2-oxazol-4-yl)-1H-1,2,4-triazole
N-(3-hydroxy-3-phenylpropyl)-N-methyl-2-(phenylamino)pyrimidine-5-carboxamide
3-{4-[1-(piperidin-1-yl)ethyl]phenyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-2-(2,5-dioxoimidazolidin-1-yl)acetamide
methyl 6-{[(2-methoxy-2-oxoethyl)(methyl)amino]methyl}-3-(5-methylthiophene-2-amido)thieno[2,3-b]pyridine-2-carboxylate
1-[(2-fluorophenyl)methyl]-N-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
(2S,4R)-N-[2-(3-fluorophenyl)ethyl]-4-[(4-fluorophenyl)sulfanyl]-1-(pyridin-2-ylmethyl)pyrrolidine-2-carboxamide
2-[2-(1-{5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carbonyl}piperidin-2-yl)ethyl]pyridine
{3-[(2-fluorophenyl)methyl]-1-[4-(trifluoromethyl)pyrimidin-2-yl]piperidin-3-yl}methanol
4-[4-(azepan-1-yl)piperidin-1-yl]-5-methylpyrimidin-2-amine
2-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propane-1,3-diol
methyl 3-(2-methylbenzoyl)-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-{3-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-3-oxopropyl}piperidin-2-one
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}ethan-1-one
benzyl (1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
(2E)-N-{[4-benzyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-3-(2-chlorophenyl)prop-2-enamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}morpholine-2-carboxamide
2-[2-benzyl-4-(3-methoxyphenyl)-5-oxopiperazin-1-yl]-N-(propan-2-yl)acetamide
1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-3-(pyridin-2-yl)propan-1-one
1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
N-[(4-fluorophenyl)methyl]-7-methyl-N-(oxolan-2-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
1-[(1-{6-[(2-hydroxyethyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
6-(4-methoxyphenyl)-3-{3-[(methylsulfanyl)methyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2-amino-6-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-4-(trimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-[3-(4-chlorophenyl)propyl]-1,1-dioxo-1λ6-thiolane-3-carboxamide
methyl 3-(3-chlorobenzamido)-6-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate