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(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-benzyl-4-({[3-(benzyloxy)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}propanamide
1-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(pyridin-4-ylmethyl)-1,4-diazepane
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-indole-6-carboxamide
(1S,5R)-6-(2-methoxyethyl)-3-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{1-[2-(propylsulfanyl)phenyl]-1H-imidazol-2-yl}pyridine
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
2-{4-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]piperidin-1-yl}acetamide
3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]propanamide
2-(3-hydroxypropyl)-8-(4-methoxybenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
1,7-dimethyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-indole-2-carboxamide
1-(cyclohexylmethyl)-3-hydroxy-3-[(4-propylpiperazin-1-yl)methyl]piperidin-2-one
3-acetyl-N-[2-(dimethylamino)-2-(4-methylphenyl)ethyl]-1H-pyrazole-5-carboxamide
6-{1-[3-(5-methyl-1,2,4-oxadiazol-3-yl)benzoyl]piperidin-4-yl}-3,4-dihydropyrimidin-4-one
(3aR,6aR)-2-[2-(4-hydroxyphenyl)ethyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]-2,8-diazaspiro[4.5]decane
N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}cyclohexanecarboxamide
5-(2-chloro-4-fluorophenyl)pyrazin-2-amine
N,N-dimethyl-2-[(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-3-yl)formamido]acetamide
2-[2-(3-methoxyphenyl)ethyl]-4-[3-(morpholine-4-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
4-benzyl-1-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)piperidin-4-ol
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-methylpyrimidine-5-carboxamide
3-(5-methylthiophen-2-yl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1H-pyrazole-5-carboxamide
5-ethyl-2-methyl-4-{3-[1-(1,3-thiazol-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
methyl[(4-methylphenyl)methyl]{[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine
4-fluoro-3-{3-methyl-5-[2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}benzene-1-sulfonamide
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-3-yl)ethyl]acetamide
N-cyclohexyl-N-methyl-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
4-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}thiomorpholine
1-[1-(2-fluorobenzoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
4-methyl-2-{3-[2-(methylsulfanyl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl}-3,4-dihydro-2H-1,4-benzoxazine
3-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridazine
6-(2,5-dimethylfuran-3-yl)-7-methyl-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-(4-hydroxyphenyl)-N-[1-(5-methylpyridin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
1-[2-(2-chlorophenyl)acetyl]-4-(cyclopropylmethyl)-1,4-diazepan-5-one
(2S,4R)-1-benzyl-N-[2-(2-fluorophenyl)ethyl]-4-[(1-propylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
(1S,9aR)-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-octahydro-1H-quinolizine
1-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-3-(thiophen-2-yl)propan-1-one
3-(azepane-1-carbonyl)-1-ethyl-N-[2-(pyridin-3-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-{[benzyl(methyl)amino]methyl}-N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-1,2-oxazole-3-carboxamide
5-[3-(hydroxymethyl)phenyl]naphthalene-1-carboxamide
[(2S)-1-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl]methanol
2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}-4-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)pyrimidine
3-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-{1-[(2-fluorophenyl)methyl]-1H-pyrazol-4-yl}urea
(4aS,7aR)-1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(1-methyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(4aS,8aR)-6-(1H-imidazol-2-ylmethyl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-[4-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)carbamoyl}amino)phenyl]-N-methylacetamide
1-[(2-methyl-1H-imidazol-4-yl)methyl]-3-phenylpiperidine
N-{5-[3-(hydroxymethyl)phenyl]-6-methylpyridin-2-yl}-2-methylpropanamide