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2-(dimethylamino)-2-(2-fluorophenyl)-1-[4-(morpholin-4-yl)piperidin-1-yl]ethan-1-one
2-(dimethylamino)-N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-methylpyrimidine-5-carboxamide
5-chloro-N-[(3R,4R)-4-hydroxypyrrolidin-3-yl]-3-phenyl-1H-indole-2-carboxamide
2-{[(1R,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-8-fluoroquinoline
1-(1-{[4-(propan-2-yl)phenyl]methyl}piperidin-4-yl)-4-(pyrrolidine-1-carbonyl)piperidine
1-ethyl-4-{[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-5-methyl-1H-pyrazole
1-(2-ethyl-2-methyl-4-oxo-3,4-dihydro-2H-1-benzopyran-6-yl)-3,3-bis(2-hydroxyethyl)urea
1-{5-methoxy-2-[(4-methoxypiperidin-1-yl)methyl]phenoxy}-3-(4-methylpiperazin-1-yl)propan-2-ol
2-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-6-methyl-1,3-benzothiazole
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1,3,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-fluoro-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-5-sulfamoylbenzamide
3-hydroxy-3-{[(2-hydroxyethyl)amino]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
1-{3-[2-methyl-4-(4-methylphenyl)piperazin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
3-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1-[5-methoxy-2-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
2-{2-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]phenoxy}acetamide
3-{[(2H-1,3-benzodioxol-5-ylmethyl)amino]methyl}-7-(methylsulfanyl)-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-2-one
3-({1-[2-(2-oxopiperidin-1-yl)acetyl]pyrrolidin-3-yl}methyl)benzoic acid
2-(4-acetyl-4-phenylpiperidin-1-yl)-N-(1-methyl-1H-pyrazol-4-yl)acetamide
N-[2-(2,4-dimethylphenoxy)ethyl]-3,4-dimethoxy-N-methylbenzamide
(1s,5s)-3,7-dimethyl-10-(pyrimidin-4-yl)-3,7,10-triazatricyclo[3.3.3.01,5]undecane
N-[(1-methyl-4-phenylpiperidin-4-yl)methyl]-1H-pyrazole-4-carboxamide
4-(1-{[5-(oxan-2-yl)thiophen-2-yl]methyl}piperidin-4-yl)pyridine
7-amino-4-(quinolin-5-yl)-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
(1R,3S,5S)-8-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane
1-(4-{[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]methyl}phenyl)imidazolidin-2-one
3-(1-hydroxy-3-methylbutan-2-yl)-1-{4-[2-(pyridin-2-yl)ethyl]phenyl}urea
methyl 4-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-4-oxobutanoate
5-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-1-ethyl-3-methyl-1H-pyrazole-5-carboxamide
methyl 4-[(2-{[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]carbamoyl}piperidin-1-yl)methyl]benzoate
2-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-2-(1H-indazol-3-yl)acetamide
(1S,4S)-2-(2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)-2-azabicyclo[2.2.1]heptane
{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl](propan-2-yl)amine
1-(3,5-dichloro-4-methylbenzoyl)azetidin-3-ol
methyl 2-(5-methyl-2-{[3-(3-methyl-1H-pyrazol-1-yl)propanamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)benzoate
4-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-amine
2-ethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]pyrimidine-5-carboxamide
3-{1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-4-yl}-1,3-oxazolidin-2-one
2-(2H-1,3-benzodioxol-5-yloxy)-1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}ethan-1-one
2-cyclopropyl-5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]pyrimidin-4-ol
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[1-(4-methoxyphenyl)propyl]-N-methylacetamide
N-({1-[2-(2-phenyl-1H-imidazol-1-yl)acetyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
2-[9-(2-methylfuran-3-carbonyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
2-(2H-1,3-benzodioxole-5-carbonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
(2S,4S)-N-ethyl-4-{[(4-fluorophenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
2-(propan-2-yl)-8-[(2-propylpyrimidin-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-cyclopentyl-N-{3-[4-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)piperidin-1-yl]phenyl}acetamide
2-{5-[3-(1H-pyrazol-1-yl)benzoyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
ethyl[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](thiophen-3-ylmethyl)amine