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2-(dimethylamino)-N-[2-(pyridin-3-yloxy)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(thiophen-3-yl)ethan-1-one
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-hydroxy-3-methoxybenzamide
methyl 3-[1-(2-oxo-1,2-dihydroquinoline-3-carbonyl)piperidin-2-yl]propanoate
N-({2-[2-(3-fluorobenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2-(1H-1,2,4-triazol-1-yl)propanamide
2-[({1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-4-yl}oxy)methyl]pyridine
N-(2,4-difluorophenyl)-3-(pyridin-4-yl)azetidine-1-carboxamide
1-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-phenylpiperidine-4-carbonitrile
N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}acetamide
N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-benzothiophene-5-carboxamide
1-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidine-1-carbonyl}cyclopropane-1-carboxamide
3-fluoro-2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
8-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
[2-({4-[(5-propylfuran-2-yl)methyl]piperazin-1-yl}methyl)phenyl]methanol
1-(benzenesulfonyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
2-[1-cyclohexyl-4-(2-methyl-5-propylpyrimidin-4-yl)piperazin-2-yl]ethan-1-ol
2-methoxy-6-(3-methylpyrazin-2-yl)-N,N-bis(propan-2-yl)benzamide
(1R,3S)-3-(2-aminoethoxy)-7-[(2,5-dimethylphenyl)methyl]-7-azaspiro[3.5]nonan-1-ol
(4aS,7aR)-1-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]-1-(2-methoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
3-[(tert-butylamino)methyl]-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
1-{2-[3-(4-chloro-2,6-dimethoxyphenyl)phenoxy]ethyl}-1H-imidazole
3-fluoro-N-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
N-[(3R,4R)-3-hydroxy-1-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]piperidin-4-yl]pyridine-2-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-ol
N-(pyridin-4-ylmethyl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
1-(2-aminoethyl)-N-cyclopropyl-N-(1,3-thiazol-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carboxamide
N-[(3R,4S)-1-acetyl-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]morpholine-4-sulfonamide
5-(3,4-difluorophenoxymethyl)-N-methyl-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
3-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
{4-[(1-ethyl-1H-indol-6-yl)methyl]morpholin-3-yl}methanol
(1R,5R)-3-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N2-{1-[2-(dimethylamino)-6-methylpyrimidin-4-yl]piperidin-4-yl}-N1-(3-methylpyridin-4-yl)ethane-1,2-diamine
({5-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-4-yl]-4-cyclopropyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
3-phenyl-N-(1-{7-[(3,4,5-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
1-[4-(2-fluorophenyl)piperazin-1-yl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
N-methyl-N-(2-methylprop-2-en-1-yl)-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
2-ethyl-4-methyl-N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-1,3-oxazole-5-carboxamide
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-[2-(cyclohex-1-en-1-yl)ethyl]acetamide
2-amino-4-[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
3-(furan-2-yl)-1-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
1-[(2E)-2-methylbut-2-en-1-yl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
N-cyclopropyl-N-{[6-(2,5-dimethoxyphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}oxolane-2-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]benzamide
N-(3-hydroxy-2,2-dimethylpropyl)-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
2-{4-[5-(aminomethyl)thiophen-2-yl]-1H-pyrazol-1-yl}-N-(3-methyl-1-phenyl-1H-pyrazol-5-yl)acetamide