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2-(2-chlorophenyl)-3-methyl-N-[3-(pyrrolidin-1-yl)propyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
(1R,2R,3S,4S)-3-amino-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}bicyclo[2.2.1]heptane-2-carboxamide
5-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-2-(methylsulfanyl)pyrimidine
2-cyclopropyl-9-(3-hydroxy-2-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
5-{[methyl({[3-(2-{4-[4-(morpholin-4-yl)benzoyl]piperazin-1-yl}ethoxy)phenyl]methyl})amino]methyl}pyrrolidin-2-one
1-(2-fluorophenyl)-5-({[2-(pyrrolidin-1-yl)ethyl]sulfanyl}methyl)-1H-1,2,4-triazole
4-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperazin-2-one
N-[1-(3-fluoro-4-methoxyphenyl)ethyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
[(3R,4R)-1-[(3,4-difluorophenyl)methyl]-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
2-{4-[(butylcarbamoyl)amino]phenyl}-2-(4-hydroxypiperidin-1-yl)acetic acid
4-[(4-hydroxy-1-methylpiperidin-4-yl)methyl]-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one
1-(4-{[(prop-2-en-1-yl)(prop-2-yn-1-yl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N-(2-{7-[(6-methylpyridin-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
5-ethyl-4-methyl-6-[4-(quinazolin-4-yl)piperazin-1-yl]pyrimidin-2-amine
(4aS,7aR)-1-{[4-(2-hydroxyethoxy)phenyl]methyl}-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(dimethylamino)-1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-1-one
5-[1-(3-phenylprop-2-ynoyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-[2-(furan-2-yl)phenyl]-1H-1,2,3-triazole
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-5-(2-methylphenyl)-1,2,4-triazin-3-amine
N-[2-(2-chlorophenyl)ethyl]-2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-(4-fluoro-2-methylphenyl)-3-[1-(quinolin-2-ylmethyl)piperidin-3-yl]propanamide
6-methyl-N-[2-(2-methylpropanesulfonyl)ethyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
2-(2-amino-9H-purin-6-yl)-N,N-bis(propan-2-yl)benzamide
N-[(2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)methyl]propanamide
4-[4-(4,6-dimethylpyrimidin-2-yl)piperazin-1-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-amine
1-(furan-2-carbonyl)-4-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-1,4-diazepane
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-hydroxypyridine-3-carboxamide
4-({2-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-N,N-dimethylpiperazine-1-carboxamide
1-ethyl-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]piperidine-4-carboxamide
3-{[4-(methoxymethyl)piperidin-1-yl]methyl}-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
5-{[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]carbamoyl}-1H-imidazole-4-carboxylic acid
N-[1-(1-cyclobutanecarbonylpiperidin-4-yl)-1H-pyrazol-5-yl]-3-phenylpropanamide
(2R,3R)-3-[methyl(3-methylbutyl)amino]-1'-(pyrimidin-2-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(2S)-2-{[4-(2-methylfuran-3-amido)phenyl]formamido}-2-phenylacetic acid
N-cyclopropyl-5-hydroxy-N-(1,3-thiazol-2-ylmethyl)pyrazine-2-carboxamide
{[2-(azocan-1-yl)pyridin-3-yl]methyl}({[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl})amine
1-(5-fluoro-2-methylbenzoyl)-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
2-ethyl-5-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-4-methyl-1,3-oxazole
4-[2-({[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]phenol
2-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-4,6-dimethylpyridine-3-carbonitrile
4-({4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
3-(1-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-imidazol-2-yl)pyridine
2-(2,4-dichlorophenoxy)-1-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]ethan-1-one
1-methyl-3-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indole
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-3-(1,2-oxazolidin-2-yl)propanamide
N4-(furan-3-ylmethyl)-N2,N2,N4,5,6-pentamethylpyrimidine-2,4-diamine
2-phenyl-1-{1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-4-yl}ethan-1-ol
9-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-[2-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-oxoethyl]-1,3-dimethylimidazolidine-2,4-dione