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2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N,N-bis(prop-2-en-1-yl)acetamide
2-oxo-2-[4-oxo-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-N-phenylacetamide
2-(3-methoxyphenoxy)-1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]ethan-1-one
[(5-ethylpyridin-2-yl)methyl]({[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})amine
3-[1-(1,3-thiazol-4-ylmethyl)piperidin-3-yl]benzoic acid
(1S,5R)-3-cyclobutanecarbonyl-6-(1H-indole-6-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(2H-1,3-benzodioxol-5-yl)-1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
2-ethyl-7-(2-methoxybenzamido)-N,1-dimethyl-N-(1H-pyrazol-5-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
1-[(4-chlorophenyl)methyl]-5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)pyrrolidin-2-one
(2,1,3-benzoxadiazol-5-ylmethyl)[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)amine
1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-N-{[3-(trifluoromethyl)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
4-[(4-fluorophenyl)methyl]-1-[6-methyl-2-(methylamino)pyrimidin-4-yl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-{2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carbonyl}-1,4-diazepane
(1R,3S)-3-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)cyclopentan-1-amine
2-({6-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-aminopyrimidin-4-yl}amino)ethan-1-ol
methyl[(3-{2-[4-(quinoline-8-sulfonyl)piperazin-1-yl]ethoxy}phenyl)methyl](thiophen-2-ylmethyl)amine
1-(2-chlorophenyl)-4-[(4-methoxy-3-{[1-(5-methylthiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine
4-({1-[5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-3-yl}methyl)morpholine
(2S,3R)-2-amino-1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-hydroxybutan-1-one
3-(2-{imidazo[2,1-b][1,3]thiazol-6-ylformamido}acetamido)propanoic acid
3-{5-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}pyridine
2-[4-(cyclopropylmethyl)-1-(3-phenylpropyl)piperazin-2-yl]ethan-1-ol
1-methyl-5-(6-oxo-1-propylpiperidine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
methyl({2-methylimidazo[1,2-a]pyridin-3-yl}methyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
2-[(oxolan-3-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-{[3-(2-fluoro-5-methoxyphenyl)phenyl]methyl}acetamide
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)pyridin-2-amine
2-{[3-(2-chlorophenyl)pyrrolidin-1-yl]methyl}-1H-imidazole
2-cyclopropyl-5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-1,3,4-oxadiazole
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}(prop-2-en-1-yl)(pyridin-2-ylmethyl)amine
(3S,5R)-1-(oxan-4-yl)-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
4-(5-{[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
(2H-1,3-benzodioxol-4-ylmethyl)(methyl)(quinolin-2-ylmethyl)amine
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-[3-(methylsulfanyl)propanoyl]-decahydro-1,6-naphthyridin-2-one
3-(3-fluoro-4-phenylbenzoyl)-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidine
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-3-[methyl(1-methylpyrrolidin-3-yl)amino]propan-1-one
3-(3-methoxyphenyl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide
(3S,4R)-N,N-dimethyl-1-(2-phenylbenzoyl)-4-propylpyrrolidin-3-amine
N,4-dimethyl-N-[(4-phenoxyphenyl)methyl]-1,3-thiazole-5-carboxamide
dimethyl({[(3S,4R)-4-(propan-2-yl)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl]sulfamoyl})amine
2-ethyl-8-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]-2,8-diazaspiro[5.5]undecan-3-one
1,3-dimethyl-N-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-[1-methyl-3-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1-(propan-2-yl)-1H-1,3-benzodiazole
3-{4-[(6-chloro-4-hydroxyquinolin-2-yl)methyl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
(2E)-N-{[3-(cycloheptyloxy)-4-methoxyphenyl]methyl}-N-cyclopropyl-3-(4-methoxyphenyl)prop-2-enamide
1-[(2-aminopyrimidin-5-yl)methyl]-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
3-[(3R,4S)-1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
N-[(2-fluoro-5-methoxyphenyl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
2-methyl-4-(1,2,3,4-tetrahydroisoquinolin-5-yl)benzoic acid
8-(oxolane-2-carbonyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one