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1,4-dimethyl-9-{[3-(prop-2-en-1-yl)-4-(prop-2-en-1-yloxy)phenyl]methyl}-1,4,9-triazaspiro[5.5]undecane
N-methyl-N-[2-({2-methylthieno[2,3-d]pyrimidin-4-yl}amino)ethyl]methanesulfonamide
N3-cyclooctyl-1-(2-methoxyethyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3-(2-methylphenyl)propanamide
(3aR,5R,6S,7aS)-2-[1-(pyridine-2-carbonyl)piperidine-4-carbonyl]-octahydro-1H-isoindole-5,6-diol
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
(3S,4R)-1-(2,3-dimethyl-1H-indole-5-carbonyl)-4-methyl-3-(2-methylpropyl)piperidin-4-ol
6-ethyl-2-methyl-N-[1-(1,3-thiazol-5-yl)propan-2-yl]quinoline-4-carboxamide
N-methyl-N-(oxolan-3-yl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
5-(benzenesulfonyl)-3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
(3S,5R)-5-[(pyridin-4-ylmethyl)carbamoyl]-1-(pyrimidin-2-yl)piperidine-3-carboxylic acid
N-methyl-5-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
(1R,5S,6R)-3-(1H-1,3-benzodiazol-2-ylmethyl)-N-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
3-chloro-1-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-oxoethyl)-5-(trifluoromethyl)-1,2-dihydropyridin-2-one
(4-phenylbutan-2-yl)({2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl})amine
N-{1-[1-(3,3-dimethylbutanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-fluorobenzamide
3-[(4aR,7aS)-4-(1-benzofuran-2-ylmethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
5-(4-cyclohexylphenyl)-3-[4-(morpholin-4-yl)piperidin-1-yl]-1,2,4-triazine
1-(dimethylamino)-2-{4-[(2,3,4-trimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-2-ol
N-[(3R,4R)-1-(6-cyanopyridin-2-yl)-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)propanamide
1-(1,3-dioxo-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindol-4-yl)-N-(2-hydroxyethyl)piperidine-4-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{2-cyclobutyl-3H-imidazo[4,5-b]pyridin-3-yl}-1-[2-(trifluoromethyl)benzenesulfonyl]piperidine
1-[2-(pyrimidin-5-yl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
1-[4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
3-{[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-5-(2-methylpropyl)-1,2,4-oxadiazole
3-(1-butyl-3-methyl-1H-1,2,4-triazol-5-yl)-1-phenylpropan-1-one
1-[4-(pyrazin-2-yl)piperazin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
1-[(1S,5R)-6-(3,5-dimethyl-1-benzofuran-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-[(1S,3R)-1-[2-(dimethylamino)ethoxy]-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
3-[2-(2,6-difluorophenyl)ethyl]-1-(furan-3-carbonyl)piperidine
2-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-N-methylpyrimidin-4-amine
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-{imidazo[1,2-a]pyridin-2-ylmethyl}-3-methyl-1,2-dihydroquinoxalin-2-one
(1S,5R)-6-(4-methoxy-2-methylbenzoyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-cycloheptyl-4-({[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}amino)pyrrolidin-2-one
2-(1,4-dithiepan-6-yl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
2-amino-4-{2-[(oxolan-2-ylmethyl)amino]pyrimidin-5-yl}-6-(propan-2-yl)pyridine-3-carbonitrile
4-(2-chlorophenyl)-3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4H-1,2,4-triazole
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
1-[(3-methoxyphenyl)methyl]-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
2-(2,2-dimethylpropyl)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-(6-methoxypyridin-3-yl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
2-ethyl-N-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]methyl}pyrimidine-5-carboxamide
(2R,3R)-1'-(4,6-dimethylpyrimidin-2-yl)-3-(1H-imidazol-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-benzyl-2-methyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
6-(2,5-dimethoxyphenyl)-2-methylquinoline
N-(3-carbamoylphenyl)-3-[(3-oxopiperazin-1-yl)methyl]benzamide
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine