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3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]propan-1-one
1-methyl-8-(2-methylquinoline-4-carbonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-(2-hydroxy-1-phenylethyl)-3-(1-methylpiperidin-4-yl)propanamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[(4-methyl-1H-imidazol-2-yl)methyl]pyrrolidine-3-carboxylic acid
N-[(2-methoxyphenyl)methyl]-3-methyl-1-propyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
N-(1-carbamoylcyclopentyl)-6-(3-fluoro-4-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
(1R,5R)-6-(2-{[(2-fluorophenyl)methyl](methyl)amino}acetyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-(3,4-difluorophenyl)-5-(3-methylfuran-2-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-3-(trifluoromethyl)pyridin-2-amine
3-(1H-indol-4-ylmethyl)-3H,4H-pyrido[2,3-d]pyrimidin-4-one
7-{[2-(2-hydroxyethyl)pyrrolidin-1-yl]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,5-dimethyl-1H-pyrazole-3-carboxamide
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-ethyl-N-(furan-2-ylmethyl)-2-oxo-N-(2-phenylethyl)-1,2-dihydropyridine-4-carboxamide
3-{4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}-1-azabicyclo[2.2.2]octane
N-[2-(2-methoxyphenyl)ethyl]-1-[(2-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
ethyl 1-(3-methoxybenzoyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
2-(dimethylamino)-2-(4-fluorophenyl)-N-[2-(1H-pyrrol-1-yl)ethyl]acetamide
(3R,4R)-1-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
1-(4-fluorophenyl)-4-(1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)piperazine
(3aS,6aS)-2-methyl-5-{4-[(methylcarbamoyl)amino]benzenesulfonyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(dimethyl-1H-1,2,4-triazol-1-yl)-N-(3-methoxypropyl)-N-{[6-(2-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}acetamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
5-(3-methoxyphenoxymethyl)-N-[(3-methyloxetan-3-yl)methyl]-1H-pyrazole-3-carboxamide
2-{[4-hydroxy-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]methyl}-6-methylquinolin-4-ol
(3-ethyl-1-{4-[(4-methylpiperazin-1-yl)methyl]benzoyl}piperidin-3-yl)methanol
1-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}-2-(1H-pyrazol-1-yl)butan-1-one
2-{5-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-3-[2-(2-methylphenyl)ethyl]piperidine
(2S,4R)-4-amino-1-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-N-ethylpyrrolidine-2-carboxamide
1-{spiro[azepane-4,2'-chromene]-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-[4-(3-fluorophenyl)phenyl]-3-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]urea
2-[(3-{5-methyl-2-[(oxolan-2-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)methyl]-1,3-benzothiazole
(4aR,7aS)-1-benzyl-4-[(4,5-dimethylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-{methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}pyridine-3-carboxamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-[3-(4-ethylphenyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl]methanol
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-(pyrrolidin-1-yl)pyrrolidine
2-{1-[(4-fluorophenyl)methyl]-4-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperazin-2-yl}ethan-1-ol
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]({[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl})methylamine
5-[(4-ethylpiperazin-1-yl)methyl]-N-(3-methoxy-2,2-dimethylpropyl)-1,2-oxazole-3-carboxamide
7-(4-fluorophenyl)-2-(1-propyl-1H-imidazol-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(pyridine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(2-methyl-4-{[(3-phenyl-1H-pyrazol-5-yl)methyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-1-[4-(thian-4-yl)piperazin-1-yl]ethan-1-one
2-(5-acetylthiophen-3-yl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methylacetamide
methyl 3-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-{4-[2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamido]phenyl}pentanamide
1-[(4-ethylphenyl)methyl]-1-(2-methoxyethyl)-3-(3-methylcinnolin-5-yl)urea
5-(1,4-oxazepane-4-carbonyl)-2-phenylpyrimidin-4-ol
2,4-dimethoxy-5-{3-[1-(pyridin-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine