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1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[4-(methoxymethyl)piperidin-1-yl]methyl}piperidin-2-one
2-methyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]imidazo[1,2-a]pyridine-6-carboxamide
1-(2,4-difluorobenzoyl)-4-(4-fluorophenyl)-1,4-diazepane
2-butyl-8-(2-ethylpyridine-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-amino-4-(5-methoxy-3-methyl-1H-indol-2-yl)-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
3-(3-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]propanamide
4-(1H-imidazol-1-yl)-1-(2-methyl-2,3-dihydro-1-benzofuran-5-carbonyl)piperidine-4-carboxylic acid
N-(2-hydroxyethyl)-3-{5-[2-(1H-pyrrol-1-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
3-(2-oxoimidazolidin-1-yl)-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]benzamide
9-[2-(7-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetyl]-1,4,9-triazaspiro[5.5]undecan-5-one
(3S,4S)-4-methyl-1-(5-propylpyrimidin-4-yl)piperidine-3,4-diol
(3R,5R)-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
2-(1-ethylpiperidin-4-yl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]acetamide
N-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-2,3-dimethylquinoxaline-6-carboxamide
2-(dimethylamino)-N-[2-(1H-imidazol-1-yl)ethyl]-6-(thiophen-2-yl)pyridine-3-carboxamide
8-(furan-3-ylmethyl)-1-(3-methylbutyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-(morpholine-4-carbonyl)piperidin-4-yl]-2-(pyridin-3-yl)acetamide
(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
methyl 6-[4-(1-hydroxy-3-methylbutyl)piperidin-1-yl]pyrimidine-4-carboxylate
N-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1-(thiophene-2-carbonyl)piperidin-3-amine
6-methoxy-N-methyl-2-oxo-N-(quinoxalin-2-ylmethyl)-1,2,3,4-tetrahydroquinoline-4-carboxamide
4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-pyrrole-2-carbonyl)piperidine
N-cyclopentyl-N'-[(4-methoxyphenyl)methyl]-N'-(oxolan-2-ylmethyl)butanediamide
N-[4-({4-[(4-methoxyphenyl)methyl]-3-oxo-6-(pyridin-3-ylmethoxy)-1,4-diazepan-1-yl}methyl)phenyl]acetamide
5-[2-(4-chloro-2-methylphenoxy)acetyl]-N-ethyl-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[1-(5-methoxypyrimidin-2-yl)piperidin-4-yl]piperidin-4-ol
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(4-methylquinolin-2-yl)piperidin-3-yl]propanoic acid
(3R,4R)-4-(hydroxymethyl)-1-[2-(phenylamino)pyrimidine-5-carbonyl]piperidin-3-ol
2-(6-methoxynaphthalen-2-yl)-4-[(4-methyl-1H-imidazol-5-yl)methyl]morpholine
4-[5-(8-chloroquinolin-2-yl)-4-phenyl-1H-imidazol-1-yl]butan-1-ol
N-cyclopropyl-1-(2-methyl-4-phenylpyrimidine-5-carbonyl)piperazine-2-carboxamide
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1,3,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{4-[(3,4-difluorophenyl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
8-[2-(2-methoxyphenyl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
2-methoxy-6-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
4-[3-(3,4-dimethylphenyl)propanoyl]-1-(2-methoxyphenyl)piperazin-2-one
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-(propan-2-yl)piperidine
3-amino-1-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
(cyclopropylmethyl)({3-methyl-1-[2-(thiomorpholin-4-yl)ethyl]-1H-pyrazol-4-yl}methyl)amine
9-methoxy-7-(5-methylthiophen-2-yl)-4-(pyridin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-[3-(3-methoxypropyl)piperidine-1-carbonyl]-4-methyl-2-(pyridin-3-yl)pyrimidine
3-ethoxy-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]propan-1-one
N-[(3R,4S)-4-cyclopropyl-1-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)pyrrolidin-3-yl]-3-methoxypropanamide
3-(5-{[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
N-ethyl-N-(4-hydroxybutyl)-3-(4-hydroxyphenyl)benzamide
ethyl 4-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-amido]piperidine-1-carboxylate
1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazine
1,3-dimethyl-2-oxo-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-2,3-dihydro-1H-1,3-benzodiazole-5-sulfonamide
1-[4-(morpholine-4-carbonyl)piperazin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
1-{2-[1-(4-methylpyridine-3-carbonyl)piperidin-4-yl]ethyl}pyrrolidin-2-one