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(3R,4R)-1-[(2-ethoxyphenyl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
4-[(2-butyl-1H-imidazol-4-yl)methyl]-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
[(3R,4R)-1-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
7-(1,3-benzothiazol-2-yl)-4-(furan-2-carbonyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(5-{[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
(2S)-1-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-2-(dipropylamino)propan-1-one
2-(4-{[7-fluoro-2-(4-methylphenyl)quinolin-3-yl]methyl}piperazin-1-yl)ethan-1-ol
3-hydroxy-1-(3-phenylpropyl)-3-[({pyrazolo[1,5-a]pyridin-3-ylmethyl}amino)methyl]piperidin-2-one
4-[(2,6-difluorophenyl)methyl]-9-methoxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-5-(naphthalen-1-yl)-1,2,4-triazin-3-amine
2-{4-[(8-methoxy-2H-chromen-3-yl)methyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
2-(4-methyl-6-{[4-(1H-pyrazol-1-yl)butan-2-yl]amino}pyrimidin-2-yl)phenol
7-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
N-[(3S,4R)-1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-propylpyrrolidin-3-yl]acetamide
N4-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-5-methylpyrimidine-2,4-diamine
2-({methyl[(3-methylthiophen-2-yl)methyl]amino}methyl)pyridine-3-carboxylic acid
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(5-ethyl-2-methylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
(2S,4R)-1-[(4-ethoxyphenyl)methyl]-N-(2-phenylethyl)-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
1-[2-(dimethylamino)ethyl]-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
(1S,5R)-6-(2-chloro-6-methylbenzenesulfonyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
5-(3-methyl-1,2,4-oxadiazol-5-yl)-2-[(1E)-pent-1-en-1-yl]pyridine
5-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{9-[(5-methylthiophen-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-1-phenylcyclopropane-1-carboxamide
(1R,5R)-6-benzyl-3-(4-methyl-1H-imidazole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
[(2,3-dimethoxyphenyl)methyl](methyl){2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
3-(3-fluorophenyl)-6-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-1-[2-(piperidin-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
5-(propane-2-sulfonyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
3-ethyl-8-{[3-(morpholin-4-ylmethyl)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{5-cyclopropyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}-2-azabicyclo[2.2.1]heptane
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-[5-(phenoxymethyl)-1,3,4-oxadiazol-2-yl]propanamide
dimethyl({[1-methyl-2-(2-methylpropyl)-7-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}-1H-1,3-benzodiazol-5-yl]sulfamoyl})amine
4-cyclopentyl-N-(4-oxo-4H-chromen-6-yl)-1,4-diazepane-1-carboxamide
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-2-phenoxyethane-1-sulfonamide
1-[4-(3-{[(2,3-dihydro-1H-inden-2-yl)amino]methyl}pyridin-2-yl)piperazin-1-yl]ethan-1-one
8-hydroxy-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methylquinoline-7-carboxamide
N-{2-[1-(but-2-yn-1-yl)-1,2,5,6-tetrahydropyridin-3-yl]ethyl}-2-chlorobenzamide
2-methoxy-N-[2-oxo-4-(pyridin-3-yl)-1,2,3,4-tetrahydroquinolin-7-yl]acetamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
5-({[1-(4-methoxybenzoyl)piperidin-4-yl]oxy}methyl)-1-methyl-1,2,3,6-tetrahydropyridine
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-3-(pyridin-2-yl)propanamide
(2S)-2-[4-(3-chloro-4-fluorophenyl)-1H-1,2,3-triazol-1-yl]-4-methylpentan-1-ol
4-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-1-(thiophen-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-chloro-N-(1-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}({imidazo[1,2-a]pyridin-3-ylmethyl})amine
N-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-N-methyloxan-4-amine
methyl (2S,4R)-1-(naphthalen-1-ylmethyl)-4-(quinoline-2-amido)pyrrolidine-2-carboxylate
2-cyclobutyl-N-(furan-2-ylmethyl)-N,1-dimethyl-7-(oxolane-2-amido)-1H-1,3-benzodiazole-5-carboxamide