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4-{[9-acetyl-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]methyl}benzonitrile
{[2-(morpholin-4-yl)pyridin-3-yl]methyl}({[5-(oxan-2-yl)furan-2-yl]methyl})amine
1-(2-methoxyphenyl)-4-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}piperazin-2-one
N-methyl-2-[(5-methyl-1,3-oxazol-4-yl)formamido]pentanamide
{4-[(4-chlorophenyl)methyl]-1-[(2-fluorophenyl)methyl]piperidin-4-yl}methanol
3-(1-benzyl-1H-pyrazol-5-yl)-1-(1,4-dioxan-2-ylmethyl)urea
(4aS,8aR)-1-(3-methoxypropyl)-6-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-decahydro-1,6-naphthyridin-2-one
2-cyclopentyl-N-{3-[4-({imidazo[1,2-a]pyridin-3-ylmethyl}amino)piperidin-1-yl]phenyl}acetamide
1-(4,6-dihydroxypyridine-3-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-{3,9-diazaspiro[5.6]dodecan-9-yl}-4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]butan-1-one
1-oxo-2-[2-(piperidin-1-yl)ethyl]-N-(thiolan-3-yl)-2,3-dihydro-1H-isoindole-5-carboxamide
3-[1-benzyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]-2-methyl-4,5,6,7-tetrahydro-1-benzofuran-4-one
1-[5-(methoxymethyl)-1,3,4-oxadiazole-2-carbonyl]-3-phenylpiperazine
4-[(4-methoxy-3-methylphenyl)methyl]-3-{2-oxo-2-[4-(pyrazin-2-yl)piperazin-1-yl]ethyl}piperazin-2-one
ethyl 5-(pyridine-3-carbonyl)-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
8-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
N-{[2-(methoxymethyl)-4-methyl-1,3-thiazol-5-yl]methyl}-6-methyl-2-(morpholin-4-yl)pyrimidin-4-amine
N-[(4-fluorophenyl)methyl]-2-(morpholin-2-yl)-N-(pyridin-4-ylmethyl)acetamide
5-({2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-2,2-dimethylthiomorpholin-3-one
1-[5-(oxolan-2-yl)thiophene-2-carbonyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
2-{2-[1-(2,3-dihydro-1-benzofuran-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
(3R)-3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1,2,3,4-tetrahydroisoquinoline
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-(dimethylamino)-2-(3-methylphenyl)acetamide
2-{5-[4-(3-methoxypropyl)piperazine-1-carbonyl]-1H-pyrazol-3-yl}phenol
8-methoxy-N-{2-[methyl(phenyl)amino]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}oxolane-2-carboxamide
4-methyl-2-[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
1-[5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(2-fluorophenoxy)piperidine
(2E)-N-{[7-(2,3-dihydro-1-benzofuran-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-phenylprop-2-enamide
8-fluoro-N-[2-(1H-imidazol-1-yl)-1-phenylethyl]quinoline-2-carboxamide
N-cyclopentyl-N-[(2,3-dimethoxyphenyl)methyl]-2-(methylamino)pyridine-4-carboxamide
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(3R)-1-[1-(4,7-dimethylquinazolin-2-yl)piperidine-3-carbonyl]pyrrolidin-3-ol
2-methoxy-5-({methyl[(methylcarbamoyl)methyl]amino}methyl)benzoic acid
3-(2,4-dichloro-3-methylphenyl)-1-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-1-methylurea
2-[({2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}amino)methyl]-6,8-dimethylquinolin-4-ol
methyl 2-[4-(cyclopropylmethyl)-5-oxo-1,4-diazepane-1-carbonyl]benzoate
N-({5-[(2,3-difluoro-4-methylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
3-cyclopropyl-4-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(1S,2R)-N1-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}-N2-propylcyclohexane-1,2-dicarboxamide
4-{3H-imidazo[4,5-b]pyridin-5-yl}-N-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
3-{2-oxo-2-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethyl}imidazolidine-2,4-dione
N-(1-{7-[(2-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
3-(4-methoxy-3,5-dimethylphenyl)-6-methylpyridazine
3-[1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]benzoic acid
N-methyl-2-(phenylamino)-N-{[2-(trifluoromethyl)phenyl]methyl}pyrimidine-5-carboxamide
1-[3-({[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
(3R,4S)-3,4-dimethyl-1-(5-propyl-1,3,4-thiadiazol-2-yl)piperidin-4-ol
[(2S,4R,5R)-5-(4-chlorophenyl)-1-ethyl-2-methyl-4-({[(2-methyl-1H-imidazol-4-yl)methyl]amino}methyl)pyrrolidin-2-yl]methanol
8-fluoro-2-{[(2-hydroxyethyl)[(trimethyl-1H-pyrazol-4-yl)methyl]amino]methyl}quinolin-4-ol