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3-[2-phenyl-2-(piperidin-1-yl)ethyl]-3,4-dihydropteridin-4-one
(2S,4S,5R)-2-ethyl-4-[(2-methoxyethyl)carbamoyl]-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
4-(1-methyl-1H-imidazol-2-yl)-1-[4-(1H-pyrrol-1-ylmethyl)benzoyl]piperidine
3-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
methyl 3-({3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]phenyl}formamido)propanoate
6-{4-[(2-hydroxy-3-methoxyphenyl)methyl]piperazin-1-yl}pyridine-3-carbonitrile
1-methyl-8-[3-(2-methyl-1H-imidazol-1-yl)propyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[(1-propyl-1H-pyrazol-4-yl)methyl]acetamide
2-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-1,3-benzodiazole-5-carboxamide
(2S,4R)-N-ethyl-1-[(5-methylfuran-2-yl)methyl]-4-[2-(morpholin-4-yl)acetamido]pyrrolidine-2-carboxamide
N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-(2-ethoxyphenyl)-N'-[3-(2-methoxyphenyl)propyl]propanediamide
1-(azocan-1-yl)-3-[2-methoxy-5-({methyl[(3-methylpyridin-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
3-(1,3-dimethyl-4-phenyl-1H-pyrazol-5-yl)-1-methyl-1-[3-(1-methyl-1H-pyrazol-4-yl)propyl]urea
1-[(2-methylphenyl)methyl]-N-[1-(pyridin-3-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
methyl 5-(7-ethoxy-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-2-hydroxybenzoate
1-(2-cyclopropylphenyl)-3-(2,2-difluoroethyl)urea
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(6-methylpyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-cyano-5-fluoro-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
N-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-1-(oxolan-2-ylmethyl)piperidin-4-amine
{1-[1-(propan-2-yl)piperidine-4-carbonyl]piperidin-4-yl}(pyridin-2-yl)methanol
2-{[4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}pyridine
1-cyclohexanecarbonyl-N-[(1r,4r)-4-hydroxycyclohexyl]pyrrolidine-2-carboxamide
1-[(4-fluorophenyl)methyl]-5-(oxane-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-methyl-3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
7-(3-chlorophenyl)-4-(4-methylpyrimidine-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3-(3-methoxyphenoxymethyl)piperidine
1-benzyl-3-(2-methylpropyl)-8-(thian-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-ethyl-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(oxolan-2-ylmethyl)propanamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-[(4-methoxyphenyl)methyl]morpholine
4-ethyl-3-{1-[2-(methylamino)-1,3-thiazole-4-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
{1-[3-(4-fluorophenyl)benzoyl]-3-[(2-methylphenyl)methyl]piperidin-3-yl}methanol
5-[2-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]-1,3,4-thiadiazol-2-amine
2-chloro-5-acetamido-N-[2-(1H-imidazol-1-yl)-1-phenylethyl]benzamide
2-(furan-2-yl)-5-(4-phenyl-1H-imidazol-5-yl)pyrimidine
N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)naphthalene-1-carboxamide
4-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-[3-(1H-imidazol-2-yl)benzoyl]-6,7-dimethoxy-1-methyl-1,2,3,4-tetrahydroisoquinoline
1-[1'-(2-amino-6-methoxypyrimidin-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
2-(6-methoxypyridin-3-yl)pyridine-4-carboxamide
N-[2-(4-{[methyl(quinolin-6-ylmethyl)amino]methyl}phenoxy)propyl]-4-(trifluoromethyl)benzamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(1-cyclopentylpiperidin-3-yl)piperazine
3-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}pyridine
3-(4-tert-butylbenzoyl)-1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidine
1-(2-{[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl](methyl)amino}ethyl)piperidin-2-one
N-cyclopropyl-3-(5-{imidazo[1,2-a]pyridine-3-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanamide
3,3-dimethyl-4-(morpholin-4-ylmethyl)-1-(5-propyl-1,3,4-thiadiazol-2-yl)piperidin-4-ol
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-phenylprop-2-ynamide
1-(2-phenylethyl)-5-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide