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3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-1-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
(3R)-3-hydroxy-N-(4-methoxy-3-propanamidophenyl)pyrrolidine-1-carboxamide
(3R,4R)-1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
1-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-2-(2H-1,2,3-triazol-2-yl)ethan-1-one
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-[3-(1H-pyrazol-1-yl)propyl]piperazine
N-(2-methoxyethyl)-4-methyl-3-[2-oxo-2-(3-oxopiperazin-1-yl)ethyl]-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-[(3R,4R)-1-(1,4-dithiepan-6-yl)-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
methyl 3-(cyclobutylmethoxy)-5-{[(5-methylpyrazin-2-yl)methyl]carbamoyl}benzoate
N-ethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1-[2-(dimethylamino)ethyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
1-methyl-3-phenyl-6-(thiolan-3-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
(5R)-5-[1-(3-methylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]pyrrolidin-2-one
N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]-2-(pyridin-2-yl)acetamide
(3S,4S)-1-[(2-aminopyridin-3-yl)methyl]-4-(2H-1,3-benzodioxol-5-yl)piperidin-3-ol
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-(3-{4-[(4-fluorophenyl)sulfanyl]piperidin-1-yl}-3-oxopropyl)pyrrolidin-2-one
1-(4-{[(2S)-1-hydroxy-4-methylpentan-2-yl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
ethyl 4-(2-methyl-4-phenylpyridine-3-amido)piperidine-1-carboxylate
1-methyl-5-(piperidin-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
N-[(2,5-difluorophenyl)methyl]-1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-[1-(2-{4-[(4-fluorophenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)-1H-pyrazol-4-yl]-2-(phenylsulfanyl)acetamide
5-(2-methylpropyl)-5-[1-(quinolin-4-ylmethyl)piperidin-4-yl]-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
2-acetyl-8-(2,3-dihydro-1H-inden-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(pyridine-2-carbonyl)-7-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinoline
3-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]urea
5-{1-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]pyrrolidin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
9-(6-chloropyridazin-3-yl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
1-(2-{4-[(2,3-dimethoxyphenyl)methyl]piperazin-1-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
5-{[4-(isoquinolin-1-yl)piperazin-1-yl]methyl}-N-propylpyrimidin-2-amine
9-(5-ethyl-1,2,4-oxadiazol-3-yl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
7-chloro-N-(2-methoxyethyl)-1-methyl-N-(thiophen-2-ylmethyl)-1H-indole-2-carboxamide
N,2-dimethyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
2-{2-[2,5-dimethoxy-4-(methylsulfanyl)phenyl]-1H-imidazol-1-yl}ethan-1-ol
(3S,4R)-4-methyl-1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-3-(2-methylpropyl)piperidin-4-ol
N-ethyl-1-[(3-methoxyphenyl)methyl]-5-(1,3-thiazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
9-[3-(1H-imidazol-1-yl)butanoyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(2-methyl-1,3-thiazol-4-yl)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)acetamide
N-{2-[1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-2-yl]ethyl}acetamide
5-({4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)-2-(thiophen-2-yl)pyrimidine
5-{[({2-chloro-9-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-3-yl}methyl)(propan-2-yl)amino]methyl}pyrrolidin-2-one
(3E)-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]pent-3-enamide
1-[(3-fluorophenyl)methyl]-4-{3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanoyl}piperazin-2-one
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
(3S,4R)-1-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
1-{2-azaspiro[4.4]nonan-2-yl}-4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butan-1-one
1-(cyclopent-1-ene-1-carbonyl)-3-(4-methoxy-2-methylbenzoyl)piperidine
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
(4aS,7aR)-N-cyclohexyl-4-(2-methoxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-{3-[(dimethylsulfamoyl)amino]phenyl}-3-methyl-3-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]urea
N-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide