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2-{1-[(3,4-difluorophenyl)carbamoyl]pyrrolidin-3-yl}benzoic acid
4-{[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-2,1,3-benzoxadiazole
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-{3-[(4-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)methyl]-2,4,6-trimethylphenyl}ethan-1-one
8-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-ethyl-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-4-methoxypiperidine
7-(cyclopropylmethyl)-2-[(4-methylpiperazin-1-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[3-(propan-2-yloxy)propyl]propanamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]oxane-2-carboxamide
N-methyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
5-[(dimethylamino)methyl]-2-(3-fluoropyridin-4-yl)phenol
4-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-3-ethyl-1H-pyrazole
methyl 8-(furan-3-ylmethyl)-1-methoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
1-methyl-N-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H-indole-6-carboxamide
1-[4-({3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
2-(pyridin-4-ylmethyl)-8-[2-(thiophen-3-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)propanamide
N-({3-methyl-7-[4-(1H-pyrazol-1-yl)butan-2-yl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-2-yl)acetamide
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-3-[3-(trifluoromethyl)benzoyl]piperidine
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-4-(pyridin-3-yl)pyrimidin-2-amine
ethyl 1-(6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carbonyl)piperidine-4-carboxylate
N-({1-[(3,5-dichloro-2-methoxyphenyl)methyl]piperidin-3-yl}methyl)acetamide
methyl (2S,4R)-1-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-4-(dimethylamino)pyrrolidine-2-carboxylate
3-fluoro-2-methoxy-N-methyl-N-(quinolin-5-ylmethyl)benzamide
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-methyl-2-phenylpropan-1-one
(1S,5R)-3-[(2,3-dimethoxyphenyl)methyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
3-(oxolan-2-yl)-7-{[4-(propan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
(3R,4S)-4-cyclopropyl-1-(2-phenylpyrimidine-5-carbonyl)pyrrolidin-3-amine
3-({[(1,3-diethyl-6-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)carbamoyl]amino}methyl)-1,2,4-oxadiazole-5-carboxamide
methyl 5-[(4-methylpentan-2-yl)amino]-3-(oxolane-3-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[4-(pyridin-2-yl)piperazin-1-yl]-3-[1-(quinolin-2-yl)piperidin-3-yl]propan-1-one
1-(1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)-2-(oxolan-2-yl)-1H-1,3-benzodiazole
(4aS,8aR)-1-(2-methylpropyl)-6-[3-(1H-pyrrol-1-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
(1R,5R)-3-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonane
(3R,4S)-3-amino-N-benzyl-4-cyclopropyl-N-methylpyrrolidine-1-sulfonamide
N-[(3S,4R)-4-propyl-1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)pyrrolidin-3-yl]methanesulfonamide
N-(5-chloro-2-methoxyphenyl)-3-[1-(3-methoxybenzoyl)piperidin-3-yl]propanamide
8-{3-[5-(4-chlorophenyl)-1H-pyrrol-2-yl]propanoyl}-2,8-diazaspiro[4.5]decan-3-one
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-({[4-(dimethylamino)phenyl]methyl}amino)-N-[2-(2-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
1-{[3-(4-chlorophenoxy)phenyl]methyl}-3-methoxypyrrolidine
methyl 2-({2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}methyl)-1,3-oxazole-4-carboxylate
6-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]quinoxaline
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}benzamide
(4aR,7aS)-1-acetyl-4-[(3,5-dimethoxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
4-({1-[1-(methoxymethyl)cyclobutanecarbonyl]piperidin-3-yl}methyl)benzoic acid
(3aR,6aS)-5-(2,1,3-benzothiadiazol-5-ylmethyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-cycloheptanecarbonylazepan-3-amine
N-{2-[(2-ethylphenyl)carbamoyl]ethyl}-3-[(2-fluorophenyl)formamido]propanamide
7-cyclohexyl-2-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2,7-diazaspiro[4.5]decan-6-one