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1-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)urea
1-({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)-3-methylpiperidine
N-(1-hydroxybutan-2-yl)-N-(pyridin-2-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}[(3-ethoxyphenyl)methyl]amino)ethan-1-ol
1-(3-methoxyphenyl)-2,2-dimethyl-4-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperazine
N-(4-fluorophenyl)-4-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperazine-2-carboxamide
2-(3-methoxypropyl)-1-{[5-(1,2-oxazol-3-yl)thiophen-2-yl]sulfonyl}piperidine
5-ethyl-2-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]pyrimidin-4-amine
1-[(4-fluorophenyl)methyl]-4-[2-methyl-2-(morpholin-4-ylmethyl)propyl]piperazin-2-one
2-methyl-N-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-[(2-fluorophenyl)methyl]-3-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-3-yl}propanamide
N-[2-(2-chlorophenyl)ethyl]-5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carboxamide
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2-(3,4,5-trimethoxyphenyl)acetamide
1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-2-(thiophen-2-yl)ethan-1-one
2-amino-4-(3,5-dichloro-2-methoxyphenyl)-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
3-({[1-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
methyl 3-{1-benzyl-3-[methyl(1,3-thiazol-4-ylmethyl)carbamoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}propanoate
N-(1-{7-[(3,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
2-{2-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}-5,6-dimethyl-2,3-dihydropyridazin-3-one
4-[(4-methyl-5-{[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]piperidine
1-(2-fluorophenyl)-4-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
N-tert-butyl-2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(2S,4R)-4-{[(2,5-difluorophenyl)methyl]amino}-N-ethyl-1-(2-methylpropyl)pyrrolidine-2-carboxamide
5-[4-(2-methoxyethoxy)piperidine-1-carbonyl]-1-(2-phenylethyl)piperidin-2-one
N-(2H-1,3-benzodioxol-4-ylmethyl)-1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(1-cyclopropylethyl)acetamide
1-acetyl-N-{2-[(2-chlorophenyl)formamido]ethyl}piperidine-3-carboxamide
(3R,4R)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
2,2-dimethylpropyl 2-[(2-methyl-1H-imidazol-4-yl)methyl]-2,7-diazaspiro[4.5]decane-7-carboxylate
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-3-ol
2-[({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]pyridine-3-carboxylic acid
N-[3-(4-chlorophenoxy)propyl]-N-methyl-4-propylpyrimidine-5-carboxamide
1-(2-{[(5-acetylpyridin-2-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)ethan-1-one
2-[(2-fluorophenyl)methyl]-6-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1,3-benzoxazole
1-methyl-3-[5-(4-methylphenyl)-1,3,4-thiadiazol-2-yl]-1-(pyrimidin-4-ylmethyl)urea
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2,6-dimethylpyrimidine-4-carboxamide
4-[1-(furan-2-ylmethyl)pyrrolidin-3-yl]-2-(2-methylphenyl)pyridine
(4aR,7aS)-1-cyclobutanecarbonyl-4-[(5-ethylpyridin-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidine-3-carboxamide
1-[9-(cyclopropylmethyl)-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-2-hydroxyethan-1-one
1-methyl-6-(propan-2-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-(4-methanesulfonylphenyl)-6-(methoxymethyl)pyrimidine
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-2-(2-methyl-1,3-thiazol-4-yl)-N-(pyridin-4-ylmethyl)acetamide
8-[(2-methyl-1,3-oxazol-4-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N,3,5-trimethyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1,2-oxazole-4-carboxamide
3-(3-methylbut-2-en-1-yl)-1-[(4-methylpiperazin-1-yl)sulfonyl]piperidine-3-carboxylic acid
N-(2-methoxy-5-{[(2-propoxypropyl)carbamoyl]amino}phenyl)acetamide
N-[(4-fluorophenyl)methyl]-1-methyl-5-{[3-(morpholin-4-yl)propyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide