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1-(2-methoxyphenyl)-4-(2-methyloxolane-2-carbonyl)piperazin-2-one
3-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]-N-(pyridin-3-yl)propanamide
(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethyl-N-(2-phenylethyl)piperidine-1-carboxamide
1-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}-4-(2-methylphenyl)piperazine
(3S)-1-[5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-methyl-1H-1,3-benzodiazol-2-yl]pyrrolidin-3-ol
1-{[(3R,4R)-1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
5-({4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-2-propylpyrimidine
(2S,4R)-4-amino-1-[1-(2,3-dihydro-1H-inden-5-yl)piperidin-4-yl]-N,N-diethylpyrrolidine-2-carboxamide
[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](methyl){[2-(methylsulfanyl)pyrimidin-5-yl]methyl}amine
(3S,4S)-4-cyclopropyl-1-[3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)propanoyl]pyrrolidine-3-carboxylic acid
5-(2-methylphenyl)-4-{1-[(5-methylthiophen-2-yl)methyl]piperidin-3-yl}-2-(pyridin-4-yl)pyrimidine
4-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]pyrimidin-2-amine
4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]-1λ6-thiomorpholine-1,1-dione
N-[3-(4-fluorophenyl)phenyl]-1-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]piperidine-3-carboxamide
1-[(3-methoxyphenyl)methyl]-6-oxo-N-(1-phenylcyclopropyl)piperidine-3-carboxamide
2-(5-{[2-(methoxymethyl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyridine
(1S,5R)-3-(pyridin-3-ylmethyl)-6-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
2-(1-{2-[methyl(phenyl)amino]ethyl}-1H-imidazol-2-yl)benzoic acid
N-tert-butyl-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
N-{1-[4-({[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}carbamoyl)phenyl]-1H-pyrazol-4-yl}furan-3-carboxamide
3-(5-acetyl-2-ethoxyphenyl)-1-[(2R)-1-hydroxy-3-(4-hydroxyphenyl)propan-2-yl]urea
1-{2-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxoethyl}pyrrolidin-2-one
6-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
(3S,4R)-1-(1-acetylpiperidine-4-carbonyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-methyl-1,2-oxazole-3-carboxamide
1-(cyclopropylmethyl)-4-[(2-phenyl-1H-imidazol-4-yl)methyl]piperazine
3-(3-chloro-1,2-oxazol-5-yl)-1-{2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
5-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-phenyl-1H-imidazole-4-carboxamide
methyl 5-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
8-({3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)quinoline
2-[4-(3-acetamidophenyl)-3,5-dimethyl-1H-pyrazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
2-[3-methyl-5-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carboxamide
1-(1-benzothiophen-2-ylmethyl)-4-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidine
N-ethyl-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]pyrrolidine-3-carboxamide
4-[4-(4-methoxyphenoxymethyl)piperidin-1-yl]-5,6-dimethylpyrimidin-2-amine
1-[4-(difluoromethoxy)-2-methylphenyl]-3-[1-(1-methyl-1H-pyrazol-4-yl)propyl]urea
(2S,4R)-4-amino-N-methyl-1-(2,3,4-trimethoxybenzoyl)pyrrolidine-2-carboxamide
2-[9-(2-hydroxyethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl]pyridine-3-carbonitrile
N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
3-acetamido-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}butanamide
N-benzyl-3-{[2-(hydroxymethyl)piperidin-1-yl]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
(3aR,7aS)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
3-[4-(dimethylamino)phenyl]-N-[2-(1H-pyrazol-4-yl)ethyl]propanamide
1-[(3,4-dimethylphenyl)methyl]-4-(1-methyl-2-oxoimidazolidine-4-carbonyl)piperazin-2-one
2-[(3,5-difluorophenyl)methyl]-8-(2-propoxyacetyl)-2,8-diazaspiro[4.5]decan-3-one
1-(3,5-dimethylphenyl)-4-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]piperazin-2-one
4-[4-(2,3-dihydro-1-benzothiophene-2-carbonyl)piperazin-1-yl]quinazoline
2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
N-(5-methanesulfonyl-2-methylphenyl)-2-phenylpyrrolidine-1-carboxamide
3-phenyl-1-(7-{[4-(pyridin-2-ylmethyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propane-1,2-dione