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2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-{[1-(2-phenylethyl)piperidin-3-yl]methyl}acetamide
2-[4-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenoxy]acetic acid
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]piperidine
methyl[(5-methylfuran-2-yl)methyl]{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
8-[3-(benzyloxy)propyl]-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
5-methyl-1-[3-(pyrrolidin-1-ylmethyl)phenyl]-1H-pyrazole-3-carboxylic acid
(3aR,6aR)-2-(cyclobutylmethyl)-5-[5-(hydroxymethyl)furan-2-carbonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)(pyridin-3-yl)methanol
2-{[3-(2-methoxyethyl)-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-1-methylpiperidine
(3S,4S)-1-({2-[3-(dimethylamino)propoxy]-3-methoxyphenyl}methyl)-4-methylpiperidine-3,4-diol
2-(4-methoxyphenyl)-5-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}pyrimidine
N-[2-(4-methoxyphenyl)ethyl]-1,5-dimethyl-N-(oxolan-2-ylmethyl)-1H-pyrazole-4-carboxamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
5-(2,4-difluorophenoxymethyl)-N-(2,3-dihydro-1H-inden-1-yl)-1,2-oxazole-3-carboxamide
2-(4-methoxy-3-methylphenyl)-4-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole
3-{3,9-diazaspiro[5.5]undecane-3-carbonyl}-1,2-dihydroquinoxalin-2-one
N-(adamantan-2-ylmethyl)-1-[(4-chlorophenyl)methyl]-6-oxopiperidine-3-carboxamide
4-[2-(4-chloro-3-methyl-1H-pyrazol-1-yl)acetyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
5-{[(5-ethyl-2-methylpyrimidin-4-yl)amino]methyl}-N,N-dimethylfuran-2-carboxamide
(3aS,6aR)-3-[2-(4-methoxyphenyl)ethyl]-5-(1H-pyrrole-2-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-(benzyloxy)-N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
9-(5,6-dimethylpyrimidin-4-yl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
3-[2-(2-fluorophenoxy)pyridin-3-yl]-1-[2-(morpholin-4-yl)ethyl]urea
1-(5-{[benzyl(methyl)amino]methyl}-1,2-oxazole-3-carbonyl)-N-ethylpyrrolidine-3-carboxamide
N-(4-{1-[2-(1H-indol-3-yl)ethyl]-1H-imidazol-2-yl}phenyl)acetamide
2-[2-({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
3-(3-fluoro-5-methylphenyl)-1-methyl-1-(oxan-2-ylmethyl)urea
3-[2-amino-4-methyl-6-(2-phenylmorpholin-4-yl)pyrimidin-5-yl]propanoic acid
[1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-3-yl]methanol
4-(1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-3-yl)benzoic acid
1-(1-methyl-1H-pyrrol-2-yl)-2-{2-[(4-methylpiperidin-1-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}ethane-1,2-dione
N-methyl-1-(oxan-4-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxamide
N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
N-methyl-2-(pyridin-3-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-5-phenoxyfuran-2-carboxamide
methyl 3-benzamido-5-[(cyclohex-3-en-1-ylmethyl)amino]-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N'-[2-(dimethylamino)ethyl]-N'-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-N,N-dimethylbutanediamide
6-cyclopentyl-2-(3-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
(1S,5R)-3-[(5-chlorothiophen-2-yl)sulfonyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2-{[1-(1-methyl-1H-imidazol-2-yl)butyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
methyl (2S)-2-{[5-(2,6-dimethylphenoxymethyl)-1,2-oxazol-3-yl]formamido}-3-methylbutanoate
(butan-2-yl)[(1,3-dimethyl-1H-pyrazol-5-yl)methyl](3-phenylprop-2-yn-1-yl)amine
3-(5-cyclobutyl-1,3,4-thiadiazol-2-yl)-1-methyl-1-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]urea
(3aS,6aR)-5-(isoquinolin-5-ylmethyl)-3-[2-(4-methoxyphenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N,1-dimethyl-3-(propan-2-yl)-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
N-ethyl-2-(3-fluorophenoxymethyl)-N-(2-hydroxyethyl)-1,3-oxazole-4-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(5-propylfuran-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[1'-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
2-cyclopentyl-9-[(2R)-2-hydroxy-2-phenylacetyl]-2,9-diazaspiro[5.5]undecan-3-one