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4-{3-methyl-1-propyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}benzonitrile
N-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazole-3-carboxamide
2-(3-hydroxypropyl)-9-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-hexyl-8-[2-(1H-imidazol-1-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}(furan-2-ylmethyl)methylamine
2-(4-fluoro-2-methoxyphenyl)quinoline
4-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(4aS,8aS)-2-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-decahydro-2,7-naphthyridin-4a-ol
(3aR,6aR)-2-methanesulfonyl-5-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-2-(3,4-dichlorophenyl)morpholine
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2-(1H-imidazol-1-yl)propanamide
N,N-dimethyl-5-[({1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}amino)methyl]-1,3-thiazol-2-amine
4-({[(2,3-difluoro-4-methoxyphenyl)methyl]amino}methyl)-6-ethyl-2H-chromen-2-one
4-{[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-2,6-dimethoxyphenol
methyl 4-(4-{[3-(4-methoxyphenoxymethyl)piperidin-1-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
1-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
4-{1-[(2-phenylpyrimidin-5-yl)methyl]piperidin-4-yl}thiomorpholine
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-5-propyl-1,2-oxazole-3-carboxamide
methyl 2-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}piperidine-1-carboxylate
2-methyl-4-{1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}pyrimidine
4-{[1-(2,4-difluorophenyl)-5-(1H-1,2,3-triazol-5-yl)-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
2-(dimethylamino)-2-(4-methylphenyl)-1-[(1s,5s)-7,10-dimethyl-3,7,10-triazatricyclo[3.3.3.01,5]undecan-3-yl]ethan-1-one
3-[4-(8-methoxyquinolin-5-yl)-3,5-dimethyl-1H-pyrazol-1-yl]propanamide
6-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-[3-oxo-3-(pyrrolidin-1-yl)propyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
4-chloro-N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylbenzamide
6-{[2-oxo-2-(pyrrolidin-1-yl)ethyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
1-[2-(methylsulfanyl)pyrimidin-4-yl]-N-[2-(pyridin-3-yloxy)propyl]piperidin-4-amine
1-cyclohexyl-4-[6-(pyridin-4-yl)pyridine-3-carbonyl]-1,4-diazepane
4-methyl-3-{pyrazolo[1,5-a]pyridin-7-yl}pyridine
1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-(4-chlorophenoxy)piperidine-4-carboxylic acid
1-methyl-4-[(2-{[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]oxy}phenyl)methyl]piperazine
8-[(2S)-2-aminopentanoyl]-3-{3-[cyclohexyl(methyl)amino]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(4-chlorophenyl)ethyl]-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-(2-methoxy-2-phenylacetyl)-N-(3-methoxypropyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
7-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
1-(5-{1H-pyrrolo[2,3-b]pyridin-4-yl}furan-2-carbonyl)piperidine
1-[2-(2,2-diphenylethyl)morpholin-4-yl]ethan-1-one
2-methyl-3-[5-(propane-1-sulfonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]-6-(trifluoromethyl)pyridine
2-(2-methoxyethoxy)-1-(3-methyl-3-phenylpiperidin-1-yl)ethan-1-one
1-(2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
N-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-5-[4-(propan-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
N-[2-(dimethylamino)ethyl]-N-methyl-3-{[1-(4-oxopentanoyl)piperidin-4-yl]oxy}benzamide
N-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]-3-(1H-indol-3-yl)propanamide
methyl (2S)-1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidine-2-carboxylate
5-cyclopropyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1,2-oxazole-3-carboxamide
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-[(3-hydroxyazetidin-1-yl)methyl]piperidin-2-one
(1S,5R)-6-benzyl-3-[3-(4-fluorophenyl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
7-[(4-fluorophenyl)methyl]-2-(pyridine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one