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3-[1-methyl-5-(2-phenoxyethyl)-1H-1,2,4-triazol-3-yl]pyridine
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-({[4-(dimethylamino)phenyl]methyl}amino)-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
N-methyl-4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]-N-[2-(oxan-2-yl)ethyl]benzamide
6-[1-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]pyrimidin-4-ol
3-[3,5-bis(trifluoromethyl)phenyl]-5,6-dimethyl-1,2-dihydropyridin-2-one
1-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}but-3-en-1-one
1-{4-[2-(3-acetylphenyl)-1H-imidazol-1-yl]phenyl}pyrrolidin-2-one
2-(1-benzofuran-5-yl)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1H-imidazole
(2S,4S)-4-amino-1-{[2-(4-methoxyphenyl)imidazo[1,2-a]pyridin-3-yl]methyl}-N-methylpyrrolidine-2-carboxamide
1-[(4aS,8aS)-7-acetyl-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-(2,5-dimethylphenyl)ethan-1-one
2-(4-chloro-3-fluorophenyl)pyridine-4-carboxamide
2-amino-4-[1-(2-hydroxyethyl)-3,5-dimethyl-1H-pyrazol-4-yl]-6-(4-hydroxyphenyl)-5-methylpyridine-3-carbonitrile
2-cyclopropyl-4-hydroxy-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}pyrimidine-5-carboxamide
6-(4-benzoylpiperidine-1-carbonyl)-2-(2-methoxyethyl)-1,3-benzoxazole
4-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyrimidin-2-amine
N-[(3-chlorophenyl)methyl]-3-{1-[(2-cyanophenyl)methyl]piperidin-4-yl}propanamide
ethyl N-[1-(3-fluorophenyl)-4-(morpholin-4-yl)-1H-indazol-3-yl]carbamate
N-methyl-5-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1H-pyrazole
N-[(5-{[1-(propan-2-yl)piperidin-4-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]cyclobutanecarboxamide
5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-N-[(3-methylpyridin-2-yl)methyl]pyridin-2-amine
N-methyl-2-(2-methyl-1H-imidazol-1-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
3-(4-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-2,5-dimethylpyrazine
N-{2-[cyclopentyl(methyl)amino]ethyl}-3-(4-hydroxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
(2-methoxyethyl)({[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl})methylamine
2-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[3-(methylsulfanyl)propyl]benzamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(5-methylthiophen-2-yl)methyl]piperidine-3-carboxamide
N-{2-[(4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}phenyl)formamido]ethyl}acetamide
2-(4-methyl-2-phenyl-1H-imidazol-1-yl)-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
N-(cyclopropylmethyl)-N-(2-methoxyethyl)-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-[(3-methylquinoxalin-2-yl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
5-{1-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
3-(4-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-1-yl)-1,2-dihydropyrazin-2-one
[(5-{1-[(1,4-dimethylpiperidin-4-yl)methyl]piperidin-4-yl}-4-ethyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
methyl 2-{[(5-oxo-1-phenylpyrrolidin-3-yl)amino]methyl}-1,3-oxazole-4-carboxylate
(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-2-(3-phenoxypropyl)-decahydroisoquinoline
N-[3-(cyclopentyloxy)propyl]-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propanamide
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-2,6-dimethylquinoline-3-carboxamide
6-ethoxy-3-{[methyl(oxan-2-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)amine
N-[(2-{2-[(dimethylsulfamoyl)amino]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
ethyl 2-(1-{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}piperidin-2-yl)acetate
1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]piperidin-4-amine
2-(2H-1,3-benzodioxol-5-yl)-1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]ethan-1-one
3-{[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzonitrile
1-[(2,6-difluorophenyl)methyl]-N-(1H-indol-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(2S,4R)-1-[(3-chlorophenyl)methyl]-N-ethyl-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
7-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-N2,N2,N4,N4-tetramethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
2-(ethylamino)-N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}pyrimidine-5-carboxamide
3-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one