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1-(methoxymethyl)-N-{[1-(2-phenylethyl)piperidin-3-yl]methyl}cyclobutane-1-carboxamide
6-(3-chlorothiophen-2-yl)-3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
1-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-3-(pyrazin-2-yl)propan-1-one
(3R,5S)-5-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]pyrrolidin-3-ol
3-[(3-chlorophenyl)methyl]-1-(3,6-dimethylpyrazin-2-yl)piperidine-3-carboxylic acid
5-(5-methyl-2-phenylfuran-3-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
6-(4-ethylphenyl)-N-methyl-N-(pyridin-3-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-{1-[(2-fluorophenyl)methyl]-1H-pyrazol-4-yl}-3-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)urea
2-[(2-fluorophenyl)methyl]-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1,3-benzoxazole-6-carboxamide
1-cyclohexyl-N-[2-(1,3-thiazol-2-yl)ethyl]piperidine-4-carboxamide
2-[3-(3-propyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]pyridine
7-fluoro-3-({methyl[3-(morpholin-4-yl)propyl]amino}methyl)-1,2-dihydroquinolin-2-one
2-oxo-2-{9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}-S-(thiophen-2-yl)ethane-1-sulfonamido
3-{2-oxo-2-[3-(4-phenylbenzoyl)piperidin-1-yl]ethyl}-3,4-dihydroquinazolin-4-one
N-[2-(2-hydroxyethoxy)ethyl]-5-[1-(1,3-thiazole-4-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
N-(3-acetylphenyl)-2,7-diazaspiro[4.5]decane-2-carboxamide
1-{3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}-2-(4-methylphenoxy)ethan-1-one
1-[(4aS,8aR)-2-oxo-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridine-6-carbonyl]cyclopropane-1-carbonitrile
2-(3-methyl-1,2-oxazol-5-yl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]acetamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-1H-indole-2-carboxamide
3-benzoyl-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperidine
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[2-(morpholin-4-yl)ethyl]amine
N-[1-(cyclohex-1-en-1-yl)ethyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
4-[(3-{2-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-2-yl]ethoxy}-4-methoxyphenyl)methyl]morpholine
8-(4-methyl-1H-imidazole-2-carbonyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
(3S,4S)-1-[1-(methoxymethyl)cyclopropanecarbonyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
2-{4-[(3-hydroxyphenyl)methyl]-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl}acetic acid
(3S,4S)-4-cyclopropyl-1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidine-3-carboxylic acid
N-({4-[(2-chloroprop-2-en-1-yl)oxy]phenyl}methyl)-4-(1H-pyrazol-1-yl)-N-(pyridin-3-ylmethyl)benzamide
5-methyl-3-{[3-(3-{pyrazolo[1,5-a]pyrimidin-3-yl}phenyl)-1H-pyrazol-1-yl]methyl}-1,2-oxazole
3,5-dimethyl-4-{[3-(4-methylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-(propan-2-yl)-1H-pyrazole
N-(3-cyclopentylpropyl)-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
5-(1-ethyl-1H-imidazol-5-yl)-1-[2-(ethylsulfanyl)ethyl]-4-phenyl-1H-imidazole
6-(benzyloxy)-4-(furan-3-carbonyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
[(4,5-dimethylfuran-2-yl)methyl]({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
3-({[4-(1H-imidazol-1-yl)phenyl]carbamoyl}(methyl)amino)-N-methylbutanamide
2-cyclopropanecarbonyl-8-(quinolin-2-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[(5-methylfuran-2-yl)methyl]propanamide
2-fluoro-5-{6-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-1,2-dihydroquinoxalin-2-one
[(3R,5R)-1-(2-methoxypyridine-4-carbonyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-ethyl-3-oxo-4-phenyl-N-(propan-2-yl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
(5S,9aS,9bS)-5-(4-ethynylphenyl)-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(3R,5S)-N-(2-hydroxyethyl)-5-(morpholin-4-ylmethyl)-1-(naphthalen-2-ylmethyl)piperidine-3-carboxamide
(2S)-1-benzyl-N-[3-(1H-indol-2-yl)phenyl]pyrrolidine-2-carboxamide
8-(2-{[(4-methoxyphenyl)methyl]carbamoyl}ethyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-butyl-1-methyl-4-[2-(1H-pyrazol-1-yl)propanoyl]piperazin-2-one
2-(3-phenyl-1,2-oxazole-4-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
N-cyclopropyl-4-[4-(1H-1,2,3,4-tetrazol-5-yl)piperidin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine