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4-(quinolin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-{3-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
2-(morpholin-4-yl)-1-[4-(quinolin-8-yl)phenyl]ethan-1-ol
(3R,4R)-1-(4-aminopyrimidin-2-yl)-4-(hydroxymethyl)piperidin-3-ol
2-{3-[(6-methylpyridin-3-yl)carbamoyl]piperazin-1-yl}-1,3-oxazole-4-carboxylic acid
6-[2-(3-cyclopentyl-1,2,4-oxadiazol-5-yl)ethyl]-2,3,4,5-tetrahydropyridazin-3-one
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-methoxypyridine-3-carboxamide
2-oxo-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-2H-pyran-5-carboxamide
ethyl 5-[(5-acetamidothiophen-2-yl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-cyclopentylpropanamide
2-[(2-chlorophenyl)methyl]-4-[3-(4-hydroxypiperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
2-[2-(dimethylamino)ethyl]-9-(4-methoxybenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
8-(5-carboxy-3-chloropyridin-2-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-4-(5-methylfuran-2-yl)benzamide
5-chloro-N-cyclopropyl-N-[(3-methoxyphenyl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
(2-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-2-yl}ethyl)dimethylamine
3-(2,6-dimethylphenoxy)-1-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}azetidine
4-[(4-ethoxyphenyl)methyl]-9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(2-{[3-methyl-4-(propan-2-yl)piperazin-1-yl]methyl}-4-(pyridin-3-yl)phenoxy)acetic acid
N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-(4-cyclohexyl-1,4-diazepan-1-yl)-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
2,3,6-trimethyl-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]quinoline-4-carboxamide
2-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}-1,2-oxazinane
2-amino-4-(3-ethyl-1H-pyrazol-5-yl)-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
2-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-4-methoxypyrimidine
N-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-2-(4-propanoylphenoxy)acetamide
benzyl 3-{[(1-methyl-6-oxo-1,6-dihydropyridin-3-yl)formamido]methyl}piperidine-1-carboxylate
2-{[1-(5-aminopyrazin-2-yl)-4-methyl-1H-1,3-benzodiazol-2-yl]methoxy}acetic acid
2-{4-[(2-ethoxyphenyl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-(3,4-dimethoxyphenyl)-1-(3,5-dimethylfuran-2-carbonyl)piperidin-3-amine
1-[2-({[2-(pyridin-4-yl)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
5-[(2,3-dihydro-1H-inden-2-yl)amino]-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl 4-{4-[2-(propan-2-ylsulfanyl)acetyl]piperazin-1-yl}benzoate
N-[1-(methoxymethyl)cyclopentyl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
2-(dimethylamino)-N-(2-hydroxyethyl)-2-(3-methylphenyl)-N-(1,3-thiazol-2-ylmethyl)acetamide
1-(2-methoxyacetyl)-N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]piperidine-4-carboxamide
(2S,4S)-1-{[4-(benzyloxy)phenyl]methyl}-N-cycloheptyl-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
1-(3-aminoazepan-1-yl)-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
2-{1-cyclopentyl-4-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]piperazin-2-yl}ethan-1-ol
(2S)-2-amino-N-[1-(3-fluorophenyl)-4-(pyridin-3-yloxy)-1H-indazol-3-yl]butanamide
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-methyl-N-[1-(pyridin-3-yl)ethyl]-1,3-oxazole-4-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N-ethyl-5-(3-phenylpiperazine-1-carbonyl)pyrimidin-2-amine
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]acetamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
6-amino-1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]hexan-1-one
1-(dimethyl-1,3-oxazole-4-carbonyl)-3-[2-(4-fluorophenyl)ethyl]piperidine
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}hexanamide
2-{[4-(2,5-dimethylphenyl)piperazin-1-yl]methyl}-4-(6-methoxypyridin-2-yl)phenol