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N-methyl-2-phenyl-N-[1-(pyridin-4-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-6-oxo-1,6-dihydropyridine-2-carboxamide
methyl 3-[(3S,4R)-1-[(3,4-difluorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoate
ethyl[3-(methylsulfanyl)butyl]{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[(1S,2R)-2-aminocyclobutyl]-3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)propanamide
N,N-dimethyl-4-{[1-methyl-3-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}aniline
N-methyl-3-(1-methylpiperidin-2-yl)-N-(1,2-oxazol-3-ylmethyl)propanamide
5-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-N-[(4-methylphenyl)methyl]-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-1-[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
N-[(3,5-difluoro-4-methoxyphenyl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
3-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
1-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(4-methylphenoxy)ethan-1-one
2-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}pyridine
methyl[2-(morpholin-4-yl)ethyl]{[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl}amine
5-(furan-3-yl)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(4-methylphenyl)pyrimidin-2-amine
(1R,3S,5S)-8-(1H-imidazol-2-ylmethyl)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octane
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl})amine
N-(1,4-oxazepan-6-ylmethyl)-9H-purin-6-amine
(1S,5R)-6-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-methyl-4-{[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]amino}pentan-2-ol
(4aR,7aS)-1-ethyl-4-(3-methoxypropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{[3-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl}benzoic acid
N-(1-{7-[(3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)oxolane-3-carboxamide
1-{7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
2-chloro-4-({[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)amino}methyl)phenol
4-[3-(1H-pyrazol-3-yl)phenyl]benzoic acid
[2-(2,3-dimethylphenoxy)ethyl][2-(pyrrolidin-1-yl)ethyl]amine
3-(2,5-dihydro-1H-pyrrole-1-carbonyl)-5-(2-methoxyphenoxymethyl)-1H-pyrazole
2-methoxy-N-[3-(pyridin-4-yl)propyl]-5-sulfamoylbenzamide
1-[5-methoxy-2-({[2-(pyridin-4-yl)ethyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
N,N-diethyl-1-{1-[(2-methylphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
N-(1-methanesulfonylpiperidin-4-yl)-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
(3S,4R)-1-(2-methoxy-5-methylbenzenesulfonyl)-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
3-({[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)amino)-1λ6-thiolane-1,1-dione
N-[(3-methoxyphenyl)methyl]-3-methyl-N-(2-methylpropyl)-4-oxo-3,4-dihydroquinazoline-7-carboxamide
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-(5-phenyl-1,3,4-thiadiazol-2-yl)piperazine-1-carboxamide
3-methoxy-1-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-1,2-dihydropyridin-2-one
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-1H-indole-3-carboxamide
1-methyl-4-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperazine-2-carboxylic acid
2-(4-methyl-1,4-diazepan-1-yl)-1-[4-(oxolan-2-ylmethyl)piperazin-1-yl]ethan-1-one
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[3-(piperidin-1-yl)propyl]acetamide
5-{[2-(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)-1H-imidazol-1-yl]methyl}thiophene-2-carboxylic acid
2-(2-fluoro-5-methoxyphenyl)-5-methyl-4-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1,3-oxazole
6-[2-(2-chlorophenoxy)acetyl]-N-{[2-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
6-methyl-5-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidine-1-carbonyl}-2-oxo-1,2-dihydropyridine-3-carbonitrile
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]benzamide
1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}azepan-2-one
N-(furan-2-ylmethyl)-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine