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2-[(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)amino]propan-1-ol
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-3-(1-methylpiperidin-2-yl)propanamide
1-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-2-one
2-(2-methyl-1,3-thiazol-4-yl)-5-(thiomorpholine-4-carbonyl)pyrimidin-4-ol
6-[(3,5-dimethoxyphenyl)methoxy]-4-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-1-(propan-2-yl)-1,4-diazepan-2-one
6-{[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
{[7-methoxy-2-(thiophen-3-yl)quinolin-3-yl]methyl}[2-(3-methoxyphenyl)ethyl]amine
2-amino-N-{2-[cyclopentyl(methyl)amino]ethyl}-N-methyl-1,3-benzothiazole-5-carboxamide
4-({4-[(3,4-difluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-4-(pyridin-3-yl)pyrimidin-2-amine
1-[1'-(5-ethyl-1,3-oxazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
4-[1-(4-ethenylbenzoyl)piperidin-4-yl]-5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidine
2-{4-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(oxolane-2-carbonyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
1-[2-(prop-2-en-1-yloxy)phenyl]-3-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]urea
N-butyl-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(propan-2-yloxy)phenyl]methyl}-2-(thiophen-3-yl)acetamide
3-[2-(4-ethylpiperidin-1-yl)ethyl]-7-methyl-3H,4H-thieno[3,2-d]pyrimidin-4-one
3-(1,3-benzothiazol-2-yl)-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}propan-1-one
1-(3-chlorophenyl)-4-[1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]piperazine
1-(3-propyl-1H-pyrazole-5-carbonyl)-4-(pyrimidin-2-yl)-1,4-diazepane
(3R,9aR)-3-benzyl-8-(thiophene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-({[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)piperidin-2-one
N-methyl-1-(2-phenylethyl)-5-[(2,2,2-trifluoroethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-amino-6-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pyrimidin-4-ol
N-methyl-N-[3-(oxolan-2-yl)propyl]-4-(piperidin-1-ylmethyl)benzamide
3-(azepane-1-carbonyl)-N,N,1-tris(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(2-methoxyethyl)-9-[2-(3-methylphenoxy)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(4-chlorophenyl)ethyl]-5-{2-[(2-methoxyethyl)amino]ethyl}pyrrolidin-2-one
1-(1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)-3-phenylpropan-1-ol
1-[1-(5-methyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
3-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-1-(4-sulfamoylphenyl)urea
1-cyclobutanecarbonyl-N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]piperidine-4-carboxamide
5-ethyl-2,3-dimethyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-[(4-ethylphenyl)methyl]-5-oxo-N-(1H-1,2,4-triazol-5-ylmethyl)pyrrolidine-3-carboxamide
N,1-dimethyl-N-[2-phenyl-1-(1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
1-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}-4,4,4-trifluorobutan-1-one
5-cyclopropyl-N-(2-hydroxyethyl)-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-methyl-1H-pyrazole-4-carboxamide
1-[(5-{1-[(2-aminopyridin-3-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-4-ol
(1S,5R)-6-(cyclobutylmethyl)-3-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(4-{[4-(1-methyl-1H-imidazol-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}phenyl)acetamide
4-(4-aminoquinolin-8-yl)-N-tert-butylbenzene-1-sulfonamide
2-ethoxy-4-({3-[4-methyl-5-(prop-2-en-1-ylsulfanyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenol
2-(ethylamino)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]pyrimidine-5-carboxamide
2-amino-7-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-{[2-(2-methoxyethyl)morpholin-4-yl]methyl}-5-methyl-1H-indole
2-[4-(3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanoyl)piperazin-1-yl]-N-(propan-2-yl)acetamide
5-fluoro-2-{5-[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}-N-methylpyrimidin-4-amine
8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-(3-methylbutyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N3-[3-(1H-indol-2-yl)phenyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide