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5-(3-methylpiperidine-1-carbonyl)-1-(2-methylpropyl)-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
N-cyclopentyl-1-{1-[(3-ethoxy-4-hydroxyphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
2-(1-benzyl-4-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl)ethan-1-ol
(2S,4S)-4-[(3-cyanopyridin-2-yl)amino]-N-ethyl-1-[(5-methylthiophen-2-yl)methyl]pyrrolidine-2-carboxamide
4-[(1-methoxybutan-2-yl)amino]-5-methyl-N-(2-methylpropyl)thieno[2,3-d]pyrimidine-6-carboxamide
N-ethyl-N-[(4-fluorophenyl)methyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
3-(2-oxo-2-{6-oxo-7-propyl-2,7-diazaspiro[4.5]decan-2-yl}ethyl)imidazolidine-2,4-dione
3-[4-(1,3-benzothiazol-2-yl)piperazine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
2-({4-phenyl-5-[(propan-2-yloxy)methyl]-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
N-[2-(4-phenylpyrimidin-2-yl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
3-[4-(2-chlorophenyl)piperazine-1-carbonyl]piperidine-1-carboxamide
2-[2-methyl-2-(morpholin-4-ylmethyl)propyl]-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[(1R,2S)-2-phenylcyclopropyl]acetamide
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[3-(1H-imidazol-1-yl)propyl]amine
N,N-dibenzyl-2-cyclopropylpyrimidine-5-carboxamide
2-(4-{[3-(4-chlorophenoxy)phenyl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
N-methyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
3-[2-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-1,3-diazinane-2,4-dione
N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[(3-chlorophenyl)methyl]-3-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]propanamide
5-{2-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methyl-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
1-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
(3S,4S)-1-(3-carbamoyl-5,6-dimethylpyridin-2-yl)-4-propylpyrrolidine-3-carboxylic acid
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-benzyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-[ethyl(4-hydroxybutyl)amino]-2-(2-methoxy-5-methylphenyl)acetic acid
6-(4-{imidazo[1,2-a]pyridine-6-carbonyl}piperazin-1-yl)pyridine-3-carbonitrile
3-[4-(3-hydroxyphenyl)piperidin-1-yl]-N-(thiophen-2-ylmethyl)propanamide
1-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
3-[2-({1-[3-(2-methylpyrimidin-4-yl)phenyl]piperidin-4-yl}amino)ethyl]-1,3-oxazolidin-2-one
6-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one
2-[5-(methoxymethyl)-1H-pyrazol-3-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(1S,5R)-1,3,3-trimethyl-6-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}-6-azabicyclo[3.2.1]octane
N-(3-methoxypropyl)-N-[(4-methylphenyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
3-{[4-(1-cyclopentanecarbonylpyrrolidin-3-yl)piperidin-1-yl]methyl}pyridine
1-(3-methoxypropyl)-3-(2-methylphenyl)-3-{2-oxo-2-[4-(thiomorpholin-4-yl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
1-[(2R)-2-amino-2-cyclohexylacetyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]morpholine-2-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-3-(2-methylpropyl)-8-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-methyl-2-(2-methyl-4-phenylpyrimidine-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(3S,9aR)-3-[(benzyloxy)methyl]-8-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-phenylacetamide
N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-3-methyl-5-propyl-1-benzofuran-2-carboxamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
5-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-N-methylthiophene-2-carboxamide
2-chloro-N-(1-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N-(1H-indazol-4-yl)-3-[(2-methyl-5-oxo-1,4-diazepan-1-yl)methyl]benzamide
(1S,5R)-3-(3-phenylpropyl)-6-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane