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(3aS,6aR)-5-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[2-(4-methoxyphenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[(2,3-dimethoxyphenyl)methyl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propane-1,3-diol
1-cycloheptyl-N-(1,2-oxazol-3-ylmethyl)-6-oxopiperidine-3-carboxamide
1-{[3-cyclopropyl-1-(2,3-dihydro-1H-inden-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-3-(1-methylpiperidin-2-yl)propanamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-N'-[2-(propan-2-yl)phenyl]butanediamide
1-(4-{1-[(1S)-1-(3-methoxyphenyl)ethyl]-1H-imidazol-2-yl}phenyl)ethan-1-one
1-(2-hydroxyethyl)-5-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-[(1-benzyl-1H-imidazol-5-yl)methyl]-4-cyclopropyl-4-methylpyrrolidin-2-one
5-cyclopropanecarbonyl-1'-(5-methoxyfuran-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-(3-hydroxy-3-methylbutyl)-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
N-(1-methoxy-2-methylpropan-2-yl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-(4-chloro-1H-pyrazol-1-yl)-1-[3-(2-ethoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
(2R,3R,6R)-3-(2-methoxyphenyl)-5-(pyridin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-[3-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1H-indazole
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1,3,5-trimethyl-1H-pyrazole-4-sulfonamide
N-(1,3-dimethyl-1H-pyrazol-4-yl)-2-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)acetamide
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-methyl-1,3-oxazole-5-carboxamide
N-[1-(4-fluorophenyl)piperidin-4-yl]-4-methyl-1H-imidazole-2-carboxamide
1-amino-N-({1-[2-methyl-2-(piperidin-1-yl)propyl]pyrrolidin-3-yl}methyl)cyclobutane-1-carboxamide
1-(3-{3-oxo-3-[4-(pyridin-2-yl)piperazin-1-yl]propyl}piperidin-1-yl)-2-phenylethane-1,2-dione
({4-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenyl}methyl)dimethylamine
N-(cyclohexylmethyl)-1-ethyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzoyl)-3,3-dimethylpiperazin-2-one
4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(propane-1-sulfonyl)piperidine
N,N-dimethyl-4-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}naphthalen-1-amine
4-[(5-chlorothiophen-2-yl)methyl]-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]-2-[4-(quinolin-6-yl)-1H-pyrazol-1-yl]acetamide
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[2-(pyridin-3-yl)acetyl]pyrrolidin-3-yl]methanesulfonamide
1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-[3-(trifluoromethyl)phenoxy]piperidine
N-(furan-2-ylmethyl)-5-[4-(4-methylphenyl)piperazine-1-carbonyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-(2-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)piperidin-2-one
[2,2-dimethyl-3-(morpholin-4-yl)propyl](methyl)(1H-pyrazol-3-ylmethyl)amine
2-(3-fluoro-4-hydroxyphenyl)-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]acetamide
6-[(diethylamino)methyl]-N-(quinolin-3-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
3-[2-(2-fluorophenyl)ethyl]-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperidine
N-ethyl-5-hydroxy-N-[2-(pyrrolidin-1-yl)ethyl]pyrazine-2-carboxamide
1-(4-methylphenyl)-4-[3-(pyridin-3-yl)propanoyl]piperazin-2-one
1-(2-methylpropyl)-4-{7-[(4-phenylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl}pyrrolidin-2-one
3-(5-methylthiophen-2-yl)-N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]-1H-pyrazole-5-carboxamide
14-(4-methyl-1H-imidazol-5-yl)-2,17-diazatetracyclo[9.8.0.03,8.013,18]nonadeca-1(19),3,5,7,11,13(18)-hexaen-16-one
[2-fluoro-5-(6-methyl-2-propylpyrimidin-4-yl)phenyl]methanol
N-[1-(pyridin-2-yl)propan-2-yl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-{[(2E)-2-methyl-3-phenylprop-2-en-1-yl]amino}pyrrolidine-2-carboxamide
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decane
1-(3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}benzoyl)azocane