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2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]pyrimidine-5-carboxamide
4-{1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]piperidine-3-carbonyl}piperazin-2-one
2-(4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)pyridine-3-carbonitrile
5-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}pyridine-2-carbonitrile
N-ethyl-5-{4-[(1-methylpiperidin-3-yl)methyl]piperazine-1-carbonyl}pyrimidin-2-amine
N-{5-[({[4-(dimethylamino)oxan-4-yl]methyl}carbamoyl)amino]-2-fluorophenyl}-2-methylpropanamide
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(1,3-thiazol-2-ylmethyl)acetamide
N-({1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)-4-methoxybenzene-1-sulfonamide
4-(1-methyl-1H-pyrazol-4-yl)-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}pyrimidin-2-amine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(1H-1,2,4-triazol-1-yl)acetamide
N-(1H-imidazol-2-ylmethyl)-N-methyl-6-(morpholin-4-yl)pyrimidin-4-amine
3-(1-butyl-1H-imidazol-2-yl)-1-[4-(difluoromethoxy)benzoyl]piperidine
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(quinolin-2-yl)piperazin-2-one
2-amino-4-(thiophen-3-yl)-6-(3,4,5-trimethoxyphenyl)pyridine-3-carbonitrile
(4aS,8aR)-2-({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)-decahydroisoquinoline
methyl 9-[(1-methylpiperidin-3-yl)methoxy]-3-(naphthalen-1-ylmethyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazole
3-[(4-fluorophenyl)formamido]-N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]propanamide
ethyl[(3-methyl-1H-pyrazol-5-yl)methyl](oxolan-2-ylmethyl)amine
5-[(4-methoxy-3-methylphenyl)methyl]-3-(2-phenylethyl)-1H-1,2,4-triazole
ethyl({[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine
2-phenoxy-1-{7-[(4-phenylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}ethan-1-one
1-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-phenylethane-1,2-dione
4-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidine-1-carbonyl]benzonitrile
2-cyclopentyl-N-[3-(4-{[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]amino}piperidin-1-yl)phenyl]acetamide
1-(3-methyl-4-oxo-3,4-dihydroquinazoline-7-carbonyl)-4-phenylpiperidine-4-carbonitrile
(4aS,7aR)-1-[(2-chlorophenyl)methyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-({4-methyl-5-[1-(6-methylpyrimidin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
5-({[(6-chloro-4-oxo-4H-chromen-3-yl)methyl](propan-2-yl)amino}methyl)pyrrolidin-2-one
5-(methoxymethyl)-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}furan-2-carboxamide
1-[(4-methanesulfonylphenyl)methyl]-2-methyl-4-(2-methylphenyl)piperazine
2-methyl-N-(prop-2-en-1-yl)-N-(pyridin-3-ylmethyl)thieno[2,3-d]pyrimidin-4-amine
N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
2-(2-phenyl-1H-imidazol-1-yl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]acetamide
8-{[4-(benzyloxy)-3-methoxyphenyl]methyl}-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
1-(1-benzothiophen-3-ylmethyl)-N-methylpiperidine-2-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1-[4-(1H-imidazol-1-yl)phenyl]piperidin-4-amine
1-{1-[(4-chlorophenyl)methyl]piperidin-4-yl}-N-cyclopropylpiperidine-3-carboxamide
N-(3-methoxyphenyl)-3-[1-(1,2,3,4-tetrahydronaphthalen-2-yl)piperidin-4-yl]propanamide
3,5-dihydroxy-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-4-methylbenzamide
(benzylsulfamoyl)[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]amine
5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-[2-(morpholin-4-yl)ethyl]piperidin-2-one
N-{[5-fluoro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methyl-1,3-thiazole-4-carboxamide
N5-cyclopentyl-N2,N2-dimethyl-5,6,7,8-tetrahydroquinazoline-2,5-diamine
5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-(3-methylbutyl)-1,2-oxazole-3-carboxamide
2-methyl-1,3-dioxo-N-[1-(2-phenylethyl)piperidin-3-yl]-2,3-dihydro-1H-isoindole-5-carboxamide
1-benzyl-4-{[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]methyl}piperidine
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-ethyl-N-[2-(pyrrolidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
ethyl({[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl})(pyridin-4-ylmethyl)amine
1'-(1-methyl-3-phenyl-1H-pyrazole-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol