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1-(2-hydroxy-4-methylpentanoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-4-(1H-pyrazol-5-yl)benzamide
N-(2-methoxyethyl)-1-[1-(6-oxo-1,6-dihydropyridazine-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
3-{2-ethyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}propanoic acid
N-[(2,3-difluorophenyl)methyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
6-cyclobutyl-2-[4-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
2-(4-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}morpholin-2-yl)ethan-1-ol
1-(furan-2-ylmethyl)-4-[2-(propylsulfanyl)pyrimidin-5-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
N,N-dimethyl-7-(pyrazine-2-carbonyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[2-(diethylamino)ethyl]-5-(methoxymethyl)-N-methyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-[(1S,2R)-2-aminocyclobutyl]-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)acetamide
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
(3S)-4-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)-3-ethylmorpholine
5-tert-butyl-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-1,3,4-oxadiazol-2-amine
2-[1-cyclopentyl-4-(quinoxalin-5-ylmethyl)piperazin-2-yl]ethan-1-ol
3-{[4-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]methyl}-1H-indole
(3aS,7aR)-5-methyl-2-(2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
2-(2,3-difluorophenyl)-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
N-(3,4-dimethylphenyl)-1-ethylpiperidin-3-amine
5-(2-phenylethyl)-5-(piperidin-4-yl)-3-(pyrazin-2-ylmethyl)imidazolidine-2,4-dione
7-chloro-4-[3-(pyridin-3-yl)azetidin-1-yl]quinoline
1-({[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)propan-2-ol
(1R,7S)-3-[(2,5-dimethylphenyl)methyl]-6-(4-methyl-1,4-diazepane-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1-ethyl-3-methyl-1H-pyrazole-5-carboxamide
5-{[(dicyclopropylmethyl)amino]methyl}-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-(2-phenylethyl)-3-propyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
N-[4-(3-chlorophenyl)phenyl]-4-ethyl-2-methyl-3-oxopiperazine-1-carboxamide
(3R,5S)-5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-1-(pyridin-4-ylmethyl)piperidine-3-carboxamide
4-[1-(3-methyl-1H-pyrazole-5-carbonyl)azetidin-3-yl]pyridine
[(3-chloro-5-fluoro-4-methoxyphenyl)methyl][(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)amine
2-methoxy-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
11-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}-4-(3-methylbutyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-[4-(3-phenylpropyl)piperazin-1-yl]-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
2-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-N-(1-methyl-1H-pyrazol-3-yl)acetamide
2-{1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-2-yl}pyridine
N,N-dimethyl-2-[(1S,5R)-6-(3-phenoxypropyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
(2S,3R)-2-amino-3-methoxy-1-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}butan-1-one
(1S,5R)-6-[(3,4-dichlorophenyl)methyl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
dimethyl[2-(2-{1-[(2R)-oxolane-2-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)ethyl]amine
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
1-[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N-{[5-(1-benzothiophen-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-methoxyacetamide
1-(furan-2-ylmethyl)-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}piperidine-3-carboxamide
N-[2-(1-{[(1-methyl-1H-pyrazol-5-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)pyridin-3-yl]cyclopropanecarboxamide
5-(methoxymethyl)-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(5-fluoro-2-methoxybenzoyl)piperidine
2-methyl-6-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-one
1-(2,5-dimethylbenzoyl)-3-(3-methoxyphenoxy)azetidine
2-(ethylamino)-N-methyl-N-[(3-methylthiophen-2-yl)methyl]pyrimidine-5-carboxamide