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N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}acetamide
2-(2-methyl-1,3-thiazol-4-yl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]acetamide
(3-{2-[1-(4-ethylbenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
N-(1H-1,3-benzodiazol-2-ylmethyl)-6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-methyl-2-{1-[(3-methyl-1-benzofuran-2-yl)methyl]-1H-imidazol-2-yl}-1H-imidazole
7-(2-hydroxy-5-methylbenzoyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-{1-[4-(1-carbamoyl-1-methylethyl)phenyl]-3,5-dimethyl-1H-pyrazol-4-yl}propanoic acid
3-{1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]azetidin-3-yl}pyridine
ethyl 2-(N-methyl-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamido)acetate
N-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
N-[1-(benzenesulfonyl)piperidin-4-yl]-3-(1-methyl-1H-pyrazol-4-yl)propanamide
5-(3-fluorophenoxymethyl)-3-[2-(4-fluorophenyl)azetidine-1-carbonyl]-1H-pyrazole
(2E)-1-{3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}-3-(thiophen-2-yl)prop-2-en-1-one
3-[(4-ethyl-1,3-thiazol-2-yl)methyl]-1-(5,7,8-trimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
(1-{3-[1-(1H-imidazol-2-ylmethyl)-4-phenyl-1H-imidazol-5-yl]phenyl}ethyl)dimethylamine
2-{4-[4-(ethylamino)pyrimidin-2-yl]-1-[(2-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-[4-(methylsulfanyl)benzoyl]piperidine
3-(3-chlorobenzoyl)-1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidine
N-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}-1H-pyrazole-4-carboxamide
1-{2-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}ethan-1-one
N-(4-fluoro-2-methylphenyl)-3-[2-(quinolin-4-yl)-1H-imidazol-1-yl]propanamide
7-(cyclohexylmethyl)-2-(1,2,3-thiadiazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-{3-[(2-fluoro-5-methylphenyl)carbamoyl]propanamido}butanoic acid
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-ol
N-[(4-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethoxy}-3-methoxyphenyl)methyl]-4-acetamido-N-[(3S)-2-oxoazepan-3-yl]benzamide
1-[(2,3-dimethoxyphenyl)methyl]-4-(pyridin-2-ylmethyl)piperazine
8-(2-methoxypyridin-3-yl)-3-methyl-2H,3H,5H,6H,7H,8H-[1,3]oxazolo[5,4-g]quinoline-2,6-dione
1,4-dimethyl-9-[4-(trifluoromethyl)pyrimidin-2-yl]-1,4,9-triazaspiro[5.5]undecane
2-methoxy-5-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)benzoic acid
2-{[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]methyl}quinolin-4-ol
N-methyl-N-[(3-methylthiophen-2-yl)methyl]-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
6-(2-methylpropyl)-2-oxo-N-(4-pentanamidophenyl)-1,2-dihydropyrimidine-4-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-(oxan-4-ylmethyl)benzamide
N-(2-hydroxyethyl)-2-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,3-benzodiazole-5-carboxamide
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[4-(2-methoxyphenyl)-1H-pyrazol-1-yl]acetamide
2-methyl-4-{4-[4-(2,2,2-trifluoroethyl)piperazine-1-carbonyl]phenyl}butan-2-ol
7-chloro-3,5-dimethyl-N-(2-oxooxolan-3-yl)-1-benzofuran-2-carboxamide
4-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
8-(3-acetylbenzoyl)-2-butyl-2,8-diazaspiro[5.5]undecan-3-one
1-methyl-3-(2-methylpropyl)-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-1H-pyrazole-5-carboxamide
methyl 1-{2-hydroxy-3-[4-({[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]propyl}piperidine-4-carboxylate
methyl 3-[(1R,9S)-5-amino-4-cyano-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-trien-3-yl]benzoate
1-{1-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]piperidin-4-yl}piperidine-3-carbonitrile
4-(5-{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]pyrrolidin-2-yl}-1,2,4-oxadiazol-3-yl)pyridine
8-[5-(hydroxymethyl)furan-2-carbonyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
(5S,9aS,9bS)-5-(2-chloro-6-fluorophenyl)-2-[(3-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[4-(4-{[2-(2,3-difluorophenyl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-5-(methoxymethyl)furan-2-carboxamide
N,2,4-trimethyl-N-[(1-phenylpyrrolidin-3-yl)methyl]pyrimidine-5-carboxamide
N-(2-phenylethyl)-1-[1-(thian-4-yl)piperidin-4-yl]piperidine-4-carboxamide