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(1S,5R)-N-[4-(furan-2-ylmethoxy)phenyl]-10-oxo-3,9-diazabicyclo[3.3.2]decane-3-carboxamide
4-ethyl-1-methyl-3-{1-[2-(pyridin-2-yl)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{1-[(2-methylphenyl)methyl]-4-(pyridin-2-ylmethyl)piperazin-2-yl}ethan-1-ol
[3-(3-phenylpropyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-yl]methanol
3-(3-{[(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)amino]methyl}-1H-indol-1-yl)propanamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[4-(4-methoxyphenyl)butan-2-yl]amine
2-chloro-4-({[(4-fluorophenyl)methyl](1-hydroxybutan-2-yl)amino}methyl)-6-methoxyphenol
N-[1-(4-chlorophenyl)ethyl]-5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}propanamide
(1S,9R)-11-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
4-(1-benzylpiperidin-4-yl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-[2-(2-fluorophenyl)-1-{1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-4-yl}ethyl]-N-methylthiophene-3-carboxamide
N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-4H-thieno[3,2-b]pyrrole-5-carboxamide
1-[(4-{2-hydroxy-3-[methyl(propan-2-yl)amino]propoxy}-3-methoxyphenyl)methyl]piperidine-4-carbonitrile
(3S)-3-ethyl-4-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)morpholine
3-{4-[6-(azepan-1-yl)pyridazin-3-yl]phenyl}propanoic acid
N-cyclopentyl-N'-[(2,5-dimethylphenyl)methyl]butanediamide
N-[1-(dimethylamino)propan-2-yl]-N'-(3-ethylphenyl)butanediamide
2-{[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-3-methyl-1H-indole
N-[2-(azepan-1-yl)-2-phenylethyl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperazin-2-one
5-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidine-1-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-6-methoxypyrimidin-4-amine
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
2-acetyl-8-[2-(4-chlorophenyl)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
7-(1,3-benzothiazol-2-yl)-4-(3-hydroxypropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-methyl-N-(pyrazin-2-ylmethyl)-1,2-oxazole-3-carboxamide
2-(3,4-dichlorophenyl)-4-(2,3-dihydro-1-benzofuran-7-carbonyl)morpholine
2-(3-{[(1,4-dithiepan-6-yl)(methyl)amino]methyl}piperidin-1-yl)ethan-1-ol
1-[1-(3,3-dimethylbutyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
benzyl[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl](cyclopropylmethyl)amine
3-{2-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
N-[(5-chloro-1H-indol-2-yl)methyl]-3-(1-methylpiperidin-2-yl)propanamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[(5-fluoro-1H-indol-2-yl)methyl]acetamide
1-(6-fluoropyridin-3-yl)-3-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}urea
(2R,3R)-3-(dimethylamino)-1'-(isoquinolin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-{[(1R,3S,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octan-8-yl]methyl}phenol
5-(3-chloropyridin-2-yl)-N-[2-(dimethylamino)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
5-methyl-N4-[3-(3-methylpiperidin-1-yl)propyl]pyrimidine-2,4-diamine
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2,5-dimethylpyrimidin-4-amine
6-chloro-2-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-2,3-dihydropyridazin-3-one
(1-{[1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methanamine
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-6-(morpholin-4-yl)pyrimidin-4-amine
5-({methyl[(3-{2-[4-(4-phenylbenzoyl)piperazin-1-yl]ethoxy}phenyl)methyl]amino}methyl)pyrrolidin-2-one
N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]-2-(thiophen-2-yl)acetamide
5-chloro-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
(3S,9aR)-8-[(2,4-dimethylphenyl)methyl]-2,3-dimethyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(2-methoxyethyl)-1-[1-(3-phenylpropanoyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
3-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1-{3-[(trifluoromethyl)sulfanyl]phenyl}urea
4-{1-[1-(2-chloro-4,5-difluorobenzoyl)piperidin-4-yl]ethyl}morpholine