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2-methoxy-N-[(3R,4S)-1-(5-methyl-1,2,4-oxadiazol-3-yl)-4-propylpyrrolidin-3-yl]acetamide
N-[4-(2-butyl-1H-imidazol-4-yl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]acetamide
6-methyl-2-{[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]amino}pyridine-3-carboxamide
4-[5-(1-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-imidazol-2-yl)pyrimidin-2-yl]morpholine
3-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane-2-carbonyl)pyridin-1-ium-1-olate
4-{[9-(2-hydroxyethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
1-{3-[2-(1H-imidazol-4-yl)-1H-imidazol-1-yl]propyl}piperidin-4-ol
1-{3-[(2,4-difluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}-2-(phenylsulfanyl)ethan-1-one
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(2-methylquinolin-8-yl)azetidine-1-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
1-(2-hydroxypyridin-3-yl)-3-[1-(3-methylphenyl)piperidin-4-yl]urea
(3S,9aR)-3-[(4-hydroxyphenyl)methyl]-8-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-ethyl-N-methyl-N-(1,2-oxazol-3-ylmethyl)-5-oxopyrrolidine-3-carboxamide
methyl[2-(oxan-4-yl)ethyl]{[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl}amine
N-[2-(2-methylphenoxy)ethyl]-1-(oxan-4-yl)piperidine-3-carboxamide
N-(2-{1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-2-yl}ethyl)acetamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyrazolo[1,5-a]pyridine-3-carboxamide
N-[(3,4-difluorophenyl)methyl]-2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-({[2-(2-hydroxyethoxy)ethyl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
(2R)-2-cyclohexyl-2-hydroxy-1-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]ethan-1-one
N-methyl-3-(piperidin-3-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)benzamide
N-[(2-fluoro-5-methoxyphenyl)methyl]-1-(pyrimidin-2-yl)piperidin-3-amine
2-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
8-[(5-ethylfuran-2-yl)methyl]-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-3,4-dihydropyrimidin-4-one
7-[(2-chloro-4-hydroxyphenyl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-{[3-(2-fluorophenoxy)azetidin-1-yl]methyl}-4-hydroxyquinoline-6-carboxamide
N-(2-hydroxyethyl)-N-methyl-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
5-(4-methanesulfonyl-1,4-diazepane-1-carbonyl)-N,N,4-trimethylpyrimidin-2-amine
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3,6-trifluorobenzamide
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
2-({[1-(4-methylpiperazin-1-yl)cyclohexyl]methyl}amino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(1-methoxybutan-2-yl)amine
{[2-(furan-2-yl)pyrimidin-5-yl]methyl}({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
(1H-imidazol-4-ylmethyl)(2-methylpropyl)(pyridin-2-ylmethyl)amine
N-[2-(2-fluorophenyl)ethyl]-5-methyl-6-(pyrrolidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
N-(1-{1-[4-(furan-2-yl)benzoyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(pyridin-4-yl)piperidin-3-yl]propanoic acid
5-(2-chloro-6-methoxyphenyl)-1H-indazol-3-amine
3-[(4-fluorophenyl)methyl]-5-[1-(2-methoxybenzoyl)piperidin-4-yl]-5-methylimidazolidine-2,4-dione
1-(2,6-dimethylpyridin-4-yl)-4-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperazine
N-(1-hydroxybutan-2-yl)-1-methyl-3-phenyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(morpholin-4-yl)butanamide
2-[4-(1-cyano-1-methylethyl)phenyl]-2-{[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}acetic acid
3-(5-{2,6-dimethylimidazo[1,2-a]pyridin-3-yl}-1,2,4-oxadiazol-3-yl)pyridazine
4-ethyl-5-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-1,3-thiazol-2-amine
3-cyclopropyl-N-[(5-methylfuran-2-yl)methyl]-1H-pyrazole-5-carboxamide
4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
3-(2-ethyl-1H-imidazol-1-yl)-N-[(4-phenyloxan-4-yl)methyl]propanamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-2-(2,4-dioxo-1,3-thiazolidin-3-yl)-N-methylacetamide