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4-{[5-(2-fluorophenyl)furan-2-yl]methyl}-1-(1H-indazol-5-yl)piperazin-2-one
N-[2-(4-methylmorpholin-2-yl)ethyl]-3-(2-oxoimidazolidin-1-yl)benzamide
10-methoxy-N-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carboxamide
8-chloro-2-{[4-(5-methylpyrimidin-4-yl)piperidin-1-yl]methyl}quinoline
1-[2-(4-fluorophenyl)piperidin-1-yl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propan-1-one
2-(dimethylamino)-8-(9H-purin-6-yl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
9-[2-(morpholin-3-yl)acetyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
3-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
N-[2-(azepan-1-yl)ethyl]-8-fluoro-N-methylquinoline-2-carboxamide
N-(2-fluoro-4-methylphenyl)-2-({7-methylpyrazolo[1,5-a]pyrimidin-6-yl}formamido)acetamide
(3S,4S)-4-(naphthalen-2-yl)-1-(1H-1,2,4-triazole-5-carbonyl)piperidin-3-ol
7-(cyclobutylmethyl)-2-{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decane
2-(3-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}phenyl)ethan-1-amine
N-[2-(azepan-1-yl)ethyl]-N-(propan-2-yl)-2,3-dihydro-1-benzofuran-7-carboxamide
methyl 3-(2-methoxy-2-phenylacetyl)-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-[4-(benzyloxy)piperidine-1-carbonyl]-1-[2-(dimethylamino)ethyl]pyrrolidin-2-one
N-(thiolan-3-yl)-9H-purin-6-amine
2-{6-chloro-3-[(4-methoxypiperidin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carbonyl}-1,2,3,4-tetrahydroisoquinoline
1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-4-(thiophen-2-ylmethyl)-1,4-diazepane
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1-benzothiophene-2-carboxamide
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-4-(4-fluorophenyl)butan-1-one
5-[1-(2,3-dihydro-1H-inden-2-yl)-1H-imidazol-2-yl]-2-(ethylsulfanyl)pyrimidine
3-{4-[1-(6-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]piperazin-1-yl}propan-1-ol
N-(1-hydroxybutan-2-yl)-N-(pyridin-3-ylmethyl)-4-(thiophen-2-yl)butanamide
3-butyl-1-methyl-4-[(3-methylthiophen-2-yl)sulfonyl]piperazin-2-one
2-ethyl-8-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
ethyl 1-[(4-methoxyphenyl)methyl]-5-[2-(morpholin-4-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(morpholin-4-yl)pyrimidine-5-carboxamide
1-{4-[(2-fluorophenyl)methyl]piperidin-1-yl}-4-(1H-imidazol-1-yl)butan-1-one
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)thian-4-amine
4-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline
5-{2-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-methyl-3-[2-({[1-(pyrazin-2-yl)propan-2-yl]carbamoyl}amino)phenyl]propanamide
(2R)-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2-hydroxypropanamide
4-(4-fluoro-2-methylphenoxy)-1-(9H-purin-6-yl)piperidine-4-carboxylic acid
2-chloro-N-(2,2-dimethyloxan-4-yl)-5-acetamido-N-methylbenzamide
4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}-N-[(3-fluorophenyl)methyl]piperidine-1-carboxamide
2-(ethoxymethyl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[1-benzyl-4-(morpholin-4-yl)-1H-indazol-3-yl]pyridine-2-carboxamide
(3S,4R)-1-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(hydroxymethyl)piperidin-3-ol
3-[5-oxo-2-(thiophen-2-ylmethyl)pyrrolidin-2-yl]-N-[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]propanamide
2-(3-{[(3S,4S)-3-hydroxy-4-(piperidin-1-yl)pyrrolidin-1-yl]methyl}phenoxy)acetamide
7-fluoro-3-methyl-2-[2-(trifluoromethyl)morpholine-4-carbonyl]-1H-indole
3-(1H-indol-3-yl)-1-(4-{1-[methyl(pyridin-4-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)propan-1-one
2-methoxy-1-{4-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]piperidin-1-yl}ethan-1-one
5-[4-(aminomethyl)piperidin-1-yl]-2-[3-(pyridin-3-yl)propyl]-2,3-dihydropyridazin-3-one
N3-cycloheptyl-4-oxo-1-(propan-2-yl)-N5-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)oxan-4-amine
(4aS,8aR)-6-[(2-butyl-1H-imidazol-4-yl)methyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one