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3-[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-1-(5-methylpyridin-3-yl)urea
1-(4-methylpiperidin-1-yl)-2-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]phenoxy}ethan-1-one
N-methyl-5-(oxolan-2-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}thiophene-2-carboxamide
1-[4-(4-methylphenyl)benzoyl]-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
[(1-benzylpyrrolidin-3-yl)methyl]({[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl})amine
4-{2-[(1-acetylpiperidin-4-yl)oxy]-5-chlorobenzoyl}piperazin-2-one
2-(pyridin-2-yl)-1-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}ethan-1-one
7-(1-methyl-1H-indole-2-carbonyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
6-(3-hydroxyazetidin-1-yl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[5-methyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidin-2-yl]-1,4-diazepane
3-(5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
4-[1-(2-methoxyethyl)piperidine-4-carbonyl]-1-(4-methylphenyl)piperazin-2-one
5-[2-(aminomethyl)-7-fluoro-2,3-dihydro-1-benzofuran-5-yl]furan-2-carboxylic acid
2-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-N-(propan-2-yl)imidazo[1,2-a]pyridine-6-carboxamide
(1R,3S)-3-[4-(2-fluoro-4-methanesulfonylphenyl)piperazine-1-carbonyl]cyclopentan-1-amine
6-(2-methylphenyl)-N-(oxolan-2-ylmethyl)-N-propylimidazo[2,1-b][1,3]thiazole-3-carboxamide
(2S,4R)-4-amino-N-(propan-2-yl)-1-(quinolin-4-ylmethyl)pyrrolidine-2-carboxamide
methyl 3-{[(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)carbamoyl]amino}benzoate
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methyl-3-(1,2-oxazinan-2-yl)propanamide
1-ethyl-5-(5-phenylpentanoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(3S,4R)-1-[(4-carboxyphenyl)methyl]-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
N-[3-methoxy-5-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-4-methyl-1,2,3,6-tetrahydropyridine-1-carboxamide
1-(6-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-3-yl)ethan-1-one
{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[2-(1H-imidazol-4-yl)ethyl]acetamide
1-[3-({[(2-chlorophenyl)methyl]amino}methyl)phenoxy]-3-[cyclohexyl(methyl)amino]propan-2-ol
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-(3,3-diphenylpiperidin-1-yl)ethan-1-one
{3-[(5-methylfuran-2-yl)methyl]-9-(pyridin-2-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
4-(1H-pyrazol-4-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]butanamide
1-[6-hydroxy-4-(3-hydroxy-4-methylbenzoyl)-1,4-diazepan-1-yl]ethan-1-one
2-[(2-methoxyethyl)(methyl)amino]-2-[2-(methylsulfanyl)phenyl]acetic acid
3-(dimethylsulfamoyl)-N-[3-(1H-imidazol-1-yl)propyl]-5-{[(3-methoxyphenyl)methyl]amino}benzamide
8-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[1-cyclohexyl-5-(1,3-thiazol-4-ylmethyl)-1H-1,2,4-triazol-3-yl](phenyl)methanol
1-({5-[(2-ethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
4-{1-butyl-5-[1-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazol-3-yl}pyridine
3-(2-phenylpropyl)-8-(pyrazine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-methyl-5-{5-[4-(5-methylfuran-2-yl)phenyl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
N-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-4-yl}-3-(4H-1,2,4-triazol-3-yl)piperidine-1-carboxamide
3-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)propanamide
N-[(2-aminopyrimidin-5-yl)methyl]-N-methyl-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
4-({[(2-ethoxyphenyl)methyl](ethyl)amino}methyl)-N-methylbenzene-1-sulfonamide
3-[(3R,4S)-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
N-methyl-N-(thiophen-2-ylmethyl)-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N,N-diethyl-4-({[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]carbamoyl}amino)-3-methylbenzamide
(4aS,8aR)-6-(2-methylpyrimidin-4-yl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
5-(propan-2-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,3,4-thiadiazol-2-amine
2-(1-{[3-(2-methylphenyl)phenyl]methyl}piperidin-2-yl)acetamide
3-{3-oxo-3-[4-(pyridin-4-yl)piperidin-1-yl]propyl}-3,4-dihydroquinazolin-4-one