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6-[(3-methoxyphenyl)methoxy]-1-(pyridin-2-ylmethyl)-4-[2-(1H-1,2,4-triazol-1-yl)propanoyl]-1,4-diazepan-2-one
2-[1-(2,2-dimethylpropyl)-4-[(2,4,6-trimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-[2-(2-chlorophenoxy)ethyl]-4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-chloro-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-5-(trifluoromethyl)benzamide
N-[(2R,3R)-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(1H-1,2,4-triazol-1-yl)acetamide
2-(2-hydroxypropyl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-(4-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperazin-1-yl)-2,5-dimethylpyrazine
(3aS,6aR)-3-[(2-methoxyphenyl)methyl]-5-[(6-methylpyridin-2-yl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-[(2-ethoxyphenyl)methyl]piperidine-4-carboxylic acid
N-(2-hydroxyethyl)-N-[(5-methylthiophen-2-yl)methyl]-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
1-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-3-methyl-3-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)urea
3-cyclopropyl-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-({3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}methyl)-2-methoxyphenol
1-(2-methoxyphenyl)-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-1H-pyrazole-4-carboxamide
2-[4-({ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-1-(morpholin-4-yl)ethan-1-one
methyl(quinolin-6-ylmethyl){[3-({1-[2-(trifluoromethyl)benzoyl]piperidin-3-yl}methoxy)phenyl]methyl}amine
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-(methylamino)pyridine-3-carboxamide
2-[1-(4-methylpyridin-3-yl)-1H-pyrazol-4-yl]ethan-1-ol
2-[4-fluoro-3-(hydroxymethyl)phenyl]-2-{methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}acetic acid
1-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-oxopyrrolidine-3-carboxylic acid
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-chloro-2-methylphenyl)urea
2-{1-[2-(3-methylphenoxy)ethyl]pyrrolidin-2-yl}pyridine
4,7,8-trimethyl-2-[4-(oxan-4-yl)piperazin-1-yl]quinoline
5-chloro-N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]-2-methylpyrimidine-4-carboxamide
4-{[3-(aminomethyl)pyrrolidin-1-yl]methyl}-N-methylbenzene-1-sulfonamide
N-(1,3-dihydroxypropan-2-yl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
1-[3-(4-{[2-(1,3-thiazol-4-yl)ethyl]amino}piperidin-1-yl)phenyl]pyrrolidin-2-one
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(3E)-N-[(4-fluorophenyl)methyl]-N-(oxolan-2-ylmethyl)pent-3-enamide
3-methyl-4-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}-1H-pyrazole
N-methyl-3-(N-methylmethanesulfonamido)-N-[(3-methylthiophen-2-yl)methyl]propanamide
N-(2-{5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazol-1-yl}ethyl)pyridine-3-carboxamide
N-cyclopropyl-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
2-(3-hydroxyphenyl)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
8-benzyl-3-ethyl-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2-methoxyethyl)-9-(5-propyl-1,3,4-thiadiazol-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(5-ethylpyridin-2-yl)methyl]-2-(3-fluorophenyl)-N-methyl-1,3-benzoxazole-5-carboxamide
ethyl 1-[(2-methoxyphenyl)carbamoyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-5-phenyl-1H-pyrazole-3-carboxamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]pyrrolidine-3-carboxylic acid
3-tert-butyl-1-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]urea
6-oxo-N-[3-(propan-2-yloxy)propyl]-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
3-methoxy-1-{[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidine
2-(dimethylamino)-7-(1,2,3,4-tetrahydroquinoline-8-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)amine
N,N-dimethyl-5-{[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}-1,3-thiazol-2-amine
3-fluoro-4-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyridine
2,6-dimethyl-8-{[3-(2-methyl-1H-imidazol-1-yl)propyl]amino}octan-2-ol
2-(1-cyclopentyl-4-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-2-yl)ethan-1-ol
1-[1-(4-fluoro-3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]but-2-yn-1-one