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4-({2-amino-3-ethyl-3H-imidazo[4,5-b]pyridin-6-yl}formamido)-N-methylbutanamide
1-cyclopentyl-N-[(1-propylpiperidin-3-yl)methyl]piperidine-4-carboxamide
2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
4-({4-methyl-5-[1-(2-propoxyethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
2-(dimethyl-1,2-oxazol-4-yl)-1-[7-(2-methylphenyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]pyrazolo[1,5-a]pyridine-7-carboxamide
N-[2-hydroxy-3-(piperazin-1-yl)propyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-{[(3-phenoxyphenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-cyano-N-({1-[(3-cyanophenyl)methyl]pyrrolidin-3-yl}methyl)benzamide
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-(pyrrolidin-1-yl)piperidine
2-{[(2-fluorophenyl)methyl](methyl)amino}-1-{2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-2-phenoxyacetamide
N-ethyl-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-[2-(2-methylphenoxy)ethyl]propanamide
4-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-1-methylpiperidine
4-(5-chloro-2-methylphenyl)-3-(2-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(3-fluorophenyl)methyl]-4-(1,2,5-thiadiazole-3-carbonyl)piperazine
4,6-dimethyl-2-{2-[(4-methylpiperazin-1-yl)methyl]phenoxy}pyridine-3-carbonitrile
1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
3-(benzyloxy)-1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
3-butyl-4-[2-(2,5-dimethoxyphenyl)acetyl]-1-methylpiperazin-2-one
N-[2-(4-fluorophenyl)ethyl]-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)[(3-methoxyphenyl)methyl]methylamine
N-[2-(3,5-dimethylphenoxy)ethyl]-N-methyl-3-(1-methylpiperidin-3-yl)propanamide
2-(2H-1,3-benzodioxol-5-yloxy)-1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]ethan-1-one
methyl 4-{7-[(2-fluorophenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-4-oxobutanoate
1-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-(cyclohex-1-en-1-yl)ethan-1-one
2-(2H-1,2,3-benzotriazol-2-yl)-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
methyl({[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl})(thiophen-3-ylmethyl)amine
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}acetamide
1-{1-[1-(4-fluoro-2-methylphenyl)piperidin-4-yl]piperidin-3-yl}-4-phenylpiperazine
3-[(3R,4S)-4-(morpholin-4-yl)-1-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]piperidin-3-yl]propan-1-ol
3-[(dimethylamino)methyl]-1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]piperidin-3-ol
6-(3-hydroxyphenyl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
1-[2-(4-chloro-2-methylphenoxy)ethyl]-4-(oxane-2-carbonyl)piperazine
N-benzyl-2-[methyl(piperidin-4-yl)amino]-N-[(6-methylpyridin-2-yl)methyl]acetamide
(2E)-N-{[3-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)-3-(thiophen-2-yl)prop-2-enamide
1-(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)piperidine-3-carboxamide
8-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[1-benzyl-5-(1-methyl-1H-pyrazol-4-yl)-1H-1,2,4-triazol-3-yl]acetamide
1-[(3-fluorophenyl)methyl]-4-(oxolane-3-carbonyl)piperazin-2-one
6-[4-(3-methylphenoxy)piperidin-1-yl]pyridine-2-carboxylic acid
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-{methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}pyridine-3-carboxamide
1-[4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]-3-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]urea
1-[(4-chlorophenyl)methyl]-N-(1H-imidazol-2-ylmethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
2-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidine-1-carbonyl]-5-methylphenol
3-{[2-(furan-3-yl)-1H-imidazol-1-yl]methyl}quinoline
1-{4-[4-(ethylamino)pyrimidin-2-yl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
5-(2-methylpropyl)-1'-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(furan-2-ylmethyl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}piperidine-3-carboxamide
N-(2-methylphenyl)-2-{4-phenyl-5-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-imidazol-1-yl}acetamide