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N-cyclopentyl-1-{1-[(4-acetamidophenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(3,5-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-{5-[(5-propylfuran-2-yl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
2-{1-[(6-methylpyridin-2-yl)methyl]-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
N-[(2R,3R)-1'-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
5-ethyl-N-{[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
5-({1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
N-cyclopentyl-3-[3-(methoxymethyl)pyrrolidine-1-carbonyl]benzene-1-sulfonamide
(1R,5S,8S)-N,N-dimethyl-3-[(2-phenylpyrimidin-5-yl)methyl]-3-azabicyclo[3.2.1]octan-8-amine
1-[2-(dimethylamino)ethyl]-5-oxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidine-3-carboxamide
1-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propane-1,2-dione
(5S,9aS,9bS)-5-(2-methoxynaphthalen-1-yl)-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-(3-fluorophenoxymethyl)-N-[2-(1,3-thiazol-4-yl)ethyl]-1H-pyrazole-3-carboxamide
N-[(2-methoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)furan-2-carboxamide
5-{[1-(2,5-difluorophenyl)cyclopropyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-[2-(dimethylamino)ethyl]-2-methyl-N-(oxolan-2-ylmethyl)-6-(piperidin-4-yl)pyrimidin-4-amine
2-(3-hydroxypropyl)-9-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
N-[(2R,4R,6S)-2-cyclohexyl-6-(5-methyl-1-propyl-1H-pyrazol-4-yl)oxan-4-yl]acetamide
2-[(2-fluorophenyl)methyl]-N-[3-(morpholin-4-yl)propyl]-1,3-benzoxazole-6-carboxamide
1-methyl-4-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperazine
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)pent-4-enamide
ethyl 4-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperazine-1-carboxylate
N,N-dimethyl-3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-(1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)-1,3-benzoxazole
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[3-(1H-imidazol-1-yl)propyl]benzamide
3-[(3R,4S)-1-(3,5-difluoro-4-methoxybenzoyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
3-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
4-(1H-imidazol-2-yl)-1-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-(1-ethyl-1H-pyrazole-5-carbonyl)-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(2S,4S)-N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-1-benzyl-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
{4-benzyl-1-[(2,5-dimethylphenyl)methyl]piperidin-4-yl}methanol
2-{1-cyclopentyl-4-[(2,3,6-trifluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
N-(1-{[(isoquinolin-5-ylmethyl)(methyl)carbamoyl]methyl}-1H-pyrazol-4-yl)-4-oxo-4-phenylbutanamide
1-(2-fluoro-4-methoxyphenyl)-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}acetamide
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
5-cyclopropyl-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
1-cyclopentyl-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidine-3-carboxamide
{[3-(4-fluorophenyl)oxolan-3-yl]methyl}(methyl)[(3-methylpyridin-2-yl)methyl]amine
N-[(3-methoxyphenyl)methyl]-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{[2-(2-methoxyethyl)morpholin-4-yl]methyl}-7-methylquinolin-2-ol
N-{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-3-azaspiro[5.5]undecan-9-amine
2-(5-carbamoyl-2-methylphenyl)-6-methoxy-N,N-bis(propan-2-yl)benzamide
1-[4-(1-benzyl-1H-pyrazole-4-carbonyl)-1,4-diazepan-1-yl]-2-methoxyethan-1-one
1-(1-{[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)-3-methylbutan-1-ol
4-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-5-(propan-2-yl)pyrimidine
3-[(2-methyl-4-phenylpyrimidin-5-yl)formamido]-N-phenylpropanamide