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5-[1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
(3E)-2-[4-(morpholin-4-yl)piperidin-1-yl]-4-phenylbut-3-enoic acid
5-(1-benzofuran-2-yl)-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1,2,4-triazin-3-amine
N-(1-methylpiperidin-4-yl)-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
1-(3-chlorophenyl)-4-[1-(2-methoxyethyl)-5-oxopyrrolidine-3-carbonyl]piperazin-2-one
(1S,5R)-3-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(3-propyl-1H-pyrazole-5-carbonyl)-4-(pyridin-2-ylmethyl)-1,4-diazepane
4-[3-(2-fluorophenyl)pyrrolidin-1-yl]pyridine
2-phenyl-N-[2-(pyridin-3-yloxy)propyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-(1,3-benzoxazol-2-ylmethyl)-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methylpropanamide
(3S,4R)-1-[5-(methoxymethyl)-1,3,4-oxadiazole-2-carbonyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
N-cyclohexyl-1,5-dimethyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-3-carboxamide
2-{4-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-2-(4,6-dimethyl-1-benzofuran-3-yl)ethan-1-one
2-[4-(2-methyl-4-phenyl-1,3-thiazole-5-carbonyl)morpholin-3-yl]acetamide
1-[(1-propyl-1H-imidazol-2-yl)methyl]-4-(pyridin-3-yl)piperazine
5-[1-(2-fluorophenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-4-methylpyrimidin-2-amine
4,6-dimethyl-3-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydropyridin-2-one
9-[6-(3-fluorophenyl)pyridine-3-carbonyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-4-carbonitrile
3-{2-[(3,5,7-trimethyl-1H-indol-2-yl)formamido]acetamido}propanoic acid
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}[(5-methylpyrazin-2-yl)methyl]amine
2-amino-4-(4-hydroxyphenyl)-6-(2-phenylethyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
methyl 1-[(3R,5S)-5-[(1,3-dihydro-2-benzofuran-5-yl)carbamoyl]-1-[(4-fluorophenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
methyl 3-[(3-fluoro-4-methoxyphenyl)methyl]-7-oxo-9-[3-(pyridin-3-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[1-(1H-indol-5-yl)ethyl]-3-(1-methyl-1H-pyrazol-4-yl)propanamide
3-(1-methyl-1H-pyrazol-4-yl)-1-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}propan-1-one
N,N,4-trimethyl-3-{[(2,4,6-trimethylpyridin-3-yl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-(1-hydroxybutan-2-yl)-3-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-1-(pyridin-3-ylmethyl)urea
5-ethyl-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylthiophene-3-carboxamide
4-[(2,2-dimethylpiperazin-1-yl)methyl]-N-(5-methyl-1,3-thiazol-2-yl)benzamide
2-amino-N-[2-(1H-indol-1-yl)ethyl]-N-methyl-1,3-benzothiazole-5-carboxamide
1-[(2-methoxypyrimidin-5-yl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
N-{4-[3-(4-chloro-1H-pyrazol-1-yl)propanamido]phenyl}pentanamide
N-[2-(2-fluorophenyl)-1-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}ethyl]-N,2-dimethylfuran-3-carboxamide
1-methyl-4-[3-(oxolan-3-yl)-5-(1H-pyrrol-3-yl)-1H-1,2,4-triazol-1-yl]piperidine
2-[1-(2,2-dimethylpropyl)-4-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperazin-2-yl]ethan-1-ol
methyl 3-(2-chloropyridine-4-carbonyl)-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
6-{2-[5-(2-fluoro-6-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyrimidin-4-ol
(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-1-[(3,4-dimethoxyphenyl)methyl]-N-(2-phenylethyl)piperidine-3-carboxamide
3-(4-fluorophenyl)-N-methyl-N-[1-(pyridin-3-yl)ethyl]-1H-pyrazole-5-carboxamide
diethyl({[3-(piperidine-1-carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]methyl})amine
pyridin-2-yl(1-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)methanol
3-[1-(3,5-dichloro-4-methylphenyl)-N-(pyridin-3-ylmethyl)formamido]propanoic acid
1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-2-(phenylsulfanyl)ethan-1-one
2-amino-6-(4-hydroxy-3-methoxyphenyl)-4-(1H-indol-5-yl)pyridine-3-carbonitrile
(2R,6R)-4-(1,4-dithiepan-6-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-[1-(3-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,5-dimethyl-1H-pyrazole