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1-(2-methoxyphenyl)-2,2-dimethyl-4-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperazine
2-(1,2-benzoxazol-3-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]acetamide
1-(2,1,3-benzoxadiazol-4-ylmethyl)-3-(cyclopropylmethyl)piperidine-3-carboxylic acid
4-chloro-3-({3-cyclopentyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1-methyl-1H-indazole
(3R,4R)-4-(azepan-1-yl)-1-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-ol
N-{[(3S,4S)-3-hydroxy-1-[2-(pyrrolidin-1-yl)acetyl]piperidin-4-yl]methyl}-2-methylbenzamide
N-({1-[(3-methyl-1-benzofuran-2-yl)methyl]pyrrolidin-3-yl}methyl)cyclopropanesulfonamide
N,N-bis(1,3-oxazol-4-ylmethyl)oxane-2-carboxamide
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)({[4-(3-methoxyphenyl)-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl})methylamine
1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(morpholin-2-yl)ethan-1-one
2,2-difluoro-1-[3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
3-{[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]amino}-2,2-dimethylpropan-1-ol
2-[3-({3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}methyl)phenoxy]acetic acid
6-[3-(2-fluorophenoxymethyl)piperidine-1-carbonyl]quinoline
4-[1-(4-fluorophenyl)cyclopropanecarbonyl]-2-(morpholin-4-ylmethyl)-1,4-oxazepane
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(4-methylphenyl)quinoline-4-carboxamide
1,6-dimethyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-2-(2,2,3,3-tetrafluoropropoxy)acetamide
4-(2,3-dimethoxyphenyl)benzamide
N-cyclopentyl-N'-[1-(3-methylpyridin-2-yl)propyl]butanediamide
N-butyl-5-fluoro-N-(furan-2-ylmethyl)-2-methoxybenzamide
N-{2-[(5,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)formamido]ethyl}-4-fluorobenzamide
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-5-(3,4-dimethylphenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
1-[1-(4-methoxyphenyl)-5-phenyl-1H-pyrazole-3-carbonyl]pyrrolidin-3-ol
2-[4-(2H-1,3-benzodioxol-4-ylmethyl)-1-methylpiperazin-2-yl]ethan-1-ol
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-[(3-fluorophenyl)methyl]piperazine
(1R,5R)-3-(5-chloro-2-fluorobenzoyl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane
ethyl 4-{[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]amino}piperidine-1-carboxylate
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2,3-diethyl-5-[(7-fluoro-2-methyl-1H-indol-3-yl)methyl]-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
5-{2-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}-1,3-dimethylimidazolidine-2,4-dione
(3aS,6aR)-5-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-(2-methanesulfonylethyl)-4-(2-methyl-1-benzofuran-7-carbonyl)piperazine
2-{6-hydroxy-4-[2-(1-methyl-1H-indol-3-yl)acetyl]-1,4-diazepan-1-yl}acetamide
5,7-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2-(2,2-dimethyloxan-4-yl)-4-{3-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
6-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-9H-purine
4-methyl-6-[2-(trifluoromethyl)morpholine-4-carbonyl]-1,3-benzothiazol-2-amine
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1H-1,3-benzodiazole-5-carboxamide
2-(dimethylamino)-1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(4-methylphenyl)ethan-1-one
2-[5-(2-methanesulfonylethyl)-3-[(2-methoxyphenyl)methyl]-1H-1,2,4-triazol-1-yl]acetic acid
methyl(1,2-oxazol-3-ylmethyl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
(3S,4S)-1-(5-chloro-2-methylbenzoyl)piperidine-3,4-diol
({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl){[2-(2-methylphenyl)pyrimidin-5-yl]methyl}amine
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
7-(2-cyclohexylethyl)-2-(pyrimidin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
5-{[1-(4-methoxy-3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-2-(methylsulfanyl)pyrimidine
2-[3-(4-fluorophenoxy)azetidin-1-yl]-4-(propan-2-yl)pyrimidine