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2-[4-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(3-phenylpropyl)piperazin-2-yl]ethan-1-ol
(1R,3S)-3-methoxy-7-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-7-azaspiro[3.5]nonan-1-ol
3-(cyclohexylamino)-N-(2,3-dihydro-1H-inden-2-yl)-5-[(propan-2-yl)sulfamoyl]benzamide
1-(oxan-4-ylmethyl)-6-(pyridin-3-ylmethoxy)-4-[3-(trifluoromethyl)benzoyl]-1,4-diazepan-2-one
4-methyl-5-oxo-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}oxolane-3-carboxamide
5-(1-cyclopropyl-5-oxopyrrolidine-3-carbonyl)-N-methyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
4-(2H-1,3-benzodioxol-5-ylmethyl)-N-(1-propyl-1H-1,2,3-triazol-4-yl)piperazine-1-carboxamide
1-cycloheptyl-N-methyl-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-(3-methoxypropyl)-1-(morpholine-4-carbonyl)piperidine-3-carboxylic acid
(4S,4aS,8aS)-4-phenyl-1-(thiophene-3-carbonyl)-decahydroquinolin-4-ol
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
1-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-4-yl)piperidin-4-ol
1-(4-tert-butylphenyl)-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-(2,4-difluorophenyl)-3-ethyl-5-(4H-1,2,4-triazol-4-ylmethyl)-1H-1,2,4-triazole
2-methyl-5-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methoxy)pyridine
N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}-3-methylthiophene-2-carboxamide
2-[4-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperazin-1-yl]-1,3-benzoxazole
N-[(3,4-dimethoxyphenyl)methyl]-4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-methylpyrimidin-2-amine
(3R,4R)-1-(3,6-dimethylpyrazin-2-yl)-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
2-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pyridine-4-carbonitrile
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-(piperidine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
methyl 3-[(2-hydroxyethyl)[(2E)-3-phenylprop-2-en-1-yl]carbamoyl]propanoate
1-[4-({methyl[(1-phenylpyrrolidin-3-yl)methyl]amino}methyl)phenyl]ethan-1-one
3-({2-[1-(4-chlorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
3-methoxy-2-[(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenol
5-(propan-2-yl)-3-{1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]pyrrolidin-2-yl}-1,2-oxazole
1-[(3-methyl-1-benzofuran-2-yl)methyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-{3-[1-(carbamoylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-6-methylpyridine-3-carboxylic acid
N3-{4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}-N1-(pyridin-3-yl)propane-1,3-diamine
N-[2-(4-fluorophenyl)-2-(piperidin-1-yl)ethyl]-2-(1H-1,2,4-triazol-1-yl)acetamide
3-methyl-4-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
2-(2,3-difluorophenyl)-N-(3,4-dimethyl-1H-pyrazol-5-yl)acetamide
1-(4-{[2-(oxolan-3-yl)-1H-imidazol-1-yl]methyl}phenyl)-1H-1,2,4-triazole
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-4-(1H-imidazol-2-yl)piperidine
1-(2-fluoro-5-methylbenzenesulfonyl)-4-hydroxypiperidine-4-carboxylic acid
methyl({[4-({1-[4-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl})(quinolin-6-ylmethyl)amine
methyl (2S,4R)-4-(dimethylamino)-1-[2-(1H-imidazol-2-yl)benzoyl]pyrrolidine-2-carboxylate
5-(2-fluorophenyl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}pyrazolo[1,5-a]pyrimidin-7-amine
2-{2-[1-methyl-3-(pyridin-3-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenoxy}acetamide
2-cyclobutyl-5-[3-(2-ethylphenoxy)azetidin-1-yl]-1,3,4-oxadiazole
methyl (2S)-1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxylate
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-{2-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
methyl 1-[(3S,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
8-(2-{[(4-fluorophenyl)methyl](methyl)amino}acetyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(2S,4S)-4-amino-N-methyl-1-[2-(2-methylpropanamido)benzoyl]pyrrolidine-2-carboxamide
(3S,4R)-1-(8-chloroquinolin-2-yl)-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
N-[(4-fluorophenyl)methyl]-3-{1-[4-(2-oxopyrrolidin-1-yl)butanoyl]piperidin-4-yl}propanamide
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetamide
{1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}(1-methyl-1H-imidazol-2-yl)methanol