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1-[1-(2,4-dimethoxybenzenesulfonyl)piperidin-4-yl]pyrrolidin-2-one
N-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-3-(methanesulfonylmethyl)piperidine-1-carboxamide
N-methyl-3-[methyl(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amino]propanamide
4-(4-methyl-1H-pyrazol-1-yl)-6-[3-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyrimidine
8-[2-(4-methylphenoxy)ethanesulfonyl]-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(methylsulfanyl)ethyl]propanamide
4-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]butanamide
3-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-2-methylphenol
1-(2-chloro-4-fluoro-5-methylphenyl)-3-[3-(2-ethyl-1H-imidazol-1-yl)propyl]urea
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-(pyridin-3-yl)piperazine
2-{1-[(2-methylphenyl)methyl]-4-(propan-2-yl)piperazin-2-yl}ethan-1-ol
(2S,4R)-4-amino-N,N-diethyl-1-(3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carbonyl)pyrrolidine-2-carboxamide
(3S,4S)-1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
2-{[(4-fluorophenyl)methyl]({[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amino}butan-1-ol
4-[1-butyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]-N-methylpyridin-2-amine
N-methyl-5-{[4-phenyl-5-(pyridin-2-yl)-1H-imidazol-1-yl]methyl}furan-2-carboxamide
2-({2-amino-6-[4-fluoro-3-(hydroxymethyl)phenyl]pyrimidin-4-yl}amino)ethan-1-ol
[3-(1H-imidazol-1-yl)propyl](pyridin-4-ylmethyl)(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
2-ethyl-N-{[4-(trifluoromethoxy)phenyl]methyl}pyrimidine-5-carboxamide
(3aS,6aS)-2-(2-hydroxyethyl)-5-[(5-methylnaphthalen-1-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-(2-hydroxyphenyl)ethan-1-one
1-{5-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-ol
(4S)-4-(propan-2-yl)-3-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-oxazolidin-2-one
2-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-3-methoxyphenol
(8R,9aS)-2-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-8-hydroxy-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
N-cyclopropyl-1-[1-(1-methyl-2-oxo-1,2-dihydropyridine-4-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
8-(2-methoxypyridine-4-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decan-3-one
N-propyl-5-{1-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1H-imidazol-2-yl}pyrimidin-2-amine
3-(2-amino-1,3-thiazol-4-yl)-1-[2-(4-chlorophenyl)morpholin-4-yl]propan-1-one
N,5-dimethyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-N-(2-methylpropyl)-1H-pyrazole-4-carboxamide
1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-methyl-2-phenoxypropan-1-one
1-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carbonyl)azocane
6-[(diethylamino)methyl]-N-(1H-imidazol-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
(2R,3R)-2-hydroxy-3-[4-(hydroxymethyl)piperidin-1-yl]-N-propyl-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-carboxamide
9-(2-hydroxyethyl)-1-methyl-4-(thiophene-3-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
3-[3-(propan-2-yloxy)benzoyl]-1-[(2,4,5-trimethoxyphenyl)methyl]piperidine
N-tert-butyl-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl)[(4-methylphenyl)methyl]amine
6-methyl-N-[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
7-(3-phenyl-1H-pyrazole-4-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2-oxopyrrolidin-1-yl)acetamide
N-[3-(3-methoxyphenyl)phenyl]-1-[3-(methylsulfanyl)propyl]piperidine-4-carboxamide
5-{1-[(3,4-difluorophenyl)methyl]-1H-imidazol-2-yl}-N-(propan-2-yl)pyrimidin-2-amine
3-({1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]piperidin-4-yl}methyl)-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2-{methyl[(1-methylpyrrolidin-2-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]acetamide
1-{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}piperidine-3-carboxamide
6-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one