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3-(5-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl)pyridine
1-[(3-hydroxy-2-oxo-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]-1,4-diazepan-5-one
2-[(1R,3S,3aS,6aR)-3-[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]-1-(hydroxymethyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]ethan-1-ol
methyl 6-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)pyridine-3-carboxylate
2-amino-4-[6-(dimethylamino)pyridin-3-yl]-6-(4-hydroxyphenyl)-5-methylpyridine-3-carbonitrile
5-{2-[(3-fluorophenyl)methoxy]phenyl}pyrazine-2-carboxylic acid
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]acetamide
3-[(2S)-2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-6-phenyl-1,2-dihydropyridin-2-one
1-(3,5-dimethylphenyl)-4-{[2-(2-hydroxyethoxy)phenyl]methyl}piperazin-2-one
1-(1H-imidazole-2-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-methyl-N-(naphthalen-1-ylmethyl)pyrimidin-2-amine
3-fluoro-N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-7-methylimidazo[1,2-a]pyridine-2-carboxamide
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N,3-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
3-[(2-methylphenyl)methyl]-1-(6-methylpyridazin-3-yl)piperidine-3-carboxylic acid
4-ethyl-N-{[1-(2-hydroxypropyl)-1,2,3,6-tetrahydropyridin-4-yl]methyl}benzamide
5-methoxy-3-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}-1H-indazole
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(1-phenylcyclopentanecarbonyl)piperidine
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-(1,2-oxazol-5-ylmethyl)benzamide
3-({4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}methyl)benzonitrile
(4aS,7aR)-4-cyclopropanecarbonyl-N-(2-methylphenyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N'-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]pentanediamide
2-{1-[(4-ethoxyphenyl)methyl]-4-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl}ethan-1-ol
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[1-(pyrazin-2-yl)piperidin-3-yl]acetamide
2-[4-(9H-fluorene-9-carbonyl)morpholin-3-yl]acetic acid
N-[3-(3-chlorophenyl)phenyl]-1-(thiophene-3-carbonyl)piperidine-4-carboxamide
1-[(1R,2R)-2-(benzyloxy)cyclopentyl]-3-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]urea
2-(1-{[1-(6-methylquinoline-4-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-ol
1-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
6-(4-methyl-3-oxopiperazin-1-yl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
1-butyl-3-cyclopropyl-5-(2,3,4-trifluorophenyl)-1H-1,2,4-triazole
1-(1-{1-[1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]propan-2-yl}-3,5-dimethyl-1H-pyrazol-4-yl)ethan-1-one
2-[2-(1H-imidazol-1-yl)ethyl]-1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)piperidine
2-(4-phenylpiperidin-1-yl)-N-(pyridin-2-ylmethyl)acetamide
2-{2-[({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
5-(3-cyclohexyl-1H-pyrazol-4-yl)-3-(1-methyl-1H-imidazol-4-yl)-1,2,4-oxadiazole
4-[1-(4-phenoxyphenyl)-1H-1,2,3,4-tetrazol-5-yl]piperazine-2-carboxylic acid
4-{5-methyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2-{2-[1-(2,6-dimethylpyridin-4-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
(1S,5R)-6-methyl-3-(2-phenylquinazolin-4-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[2-fluoro-3-(trifluoromethyl)phenyl]methyl}-2,5-dimethyl-1,3-thiazole-4-carboxamide
(3aS,6aS)-5-(3-ethoxypropanoyl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-ethyl-3-(piperidine-1-carbonyl)-5-(pyrrolidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole
5-[4-(3-methoxypropyl)piperazine-1-carbonyl]-1H-imidazole-4-carboxylic acid
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]benzamide
[(3R,4R)-1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
3-[(1-{2-[methyl(1-methylpiperidin-4-yl)amino]acetyl}pyrrolidin-3-yl)methyl]benzamide
N-{3-oxo-3-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propyl}methanesulfonamide
N-[1-(4-fluorophenyl)-4-(morpholin-4-yl)-1H-indazol-3-yl]-2-propoxyacetamide
1-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
4-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-2-phenylpiperazine