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1-cycloheptanecarbonyl-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-(1H-1,3-benzodiazol-2-ylmethyl)-5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
3-{5-[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]-4-phenyl-1H-imidazol-1-yl}propan-1-ol
1,5-dimethyl-2-phenyl-4-{[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-2,3-dihydro-1H-pyrazol-3-one
(1R,3S)-3-(2-aminoethoxy)-7-[(2,6-dichlorophenyl)methyl]-7-azaspiro[3.5]nonan-1-ol
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]propanamide
2-(cyclopropylmethyl)-N-(2,5-dimethylphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-cyclopropyl-4-{[4-(2-phenylethoxy)phenyl]methyl}piperazine-2-carboxamide
({5-[1-(isoquinolin-1-yl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
3-(3-fluorophenyl)-6-(6-hydroxypyridine-3-carbonyl)-1-[2-(piperidin-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-{1-[2-(pyridin-3-yl)acetyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
2-(2,2-dimethylpropanamido)-5-methyl-N-[2-(morpholin-4-yl)butyl]thiophene-3-carboxamide
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3,3,3-trifluoropropan-1-one
ethyl 5-{imidazo[1,2-a]pyridine-2-carbonyl}-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-{4-[5-(4-chlorophenyl)-1,2,4-triazin-3-yl]piperazin-1-yl}-N,N-dimethylacetamide
(1S,3R)-3-amino-N-[2-(2-fluorophenoxy)ethyl]-N-(2-methoxyethyl)cyclopentane-1-carboxamide
[(3R,5S)-5-(morpholin-4-ylmethyl)-1-[(4-phenylphenyl)methyl]piperidin-3-yl]methanol
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
(3aR,6aS)-5-{[4-methoxy-3-(prop-2-en-1-yl)phenyl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-oxo-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}-1,2-dihydroquinoline-4-carboxamide
ethyl 9-[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]-3-azaspiro[5.5]undecane-3-carboxylate
3-{1-[(1-propyl-1H-pyrazol-5-yl)sulfonyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
N-(isoquinolin-5-ylmethyl)-N-methyl-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
ethyl 3-({3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxyphenyl}formamido)propanoate
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}[(3,4-dimethoxyphenyl)methyl]methylamine
methyl 6-cyclohexanecarbonyl-2-{[(4-fluorophenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-{3-[cyclohexyl(methyl)amino]propyl}-8-propanoyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(1H-imidazol-4-ylmethyl)-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
7-fluoro-3-{[(2-methoxyethyl)(oxolan-2-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
2-(4-{[4-(methylamino)piperidin-1-yl]methyl}phenyl)-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
4-[(6-methylpyridin-3-yl)oxy]-1-(thiophene-3-carbonyl)piperidine-4-carboxylic acid
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[(5-methylpyrazin-2-yl)methyl]amine
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-{[3-(methylsulfanyl)phenyl]methyl}urea
4-[1-methyl-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]morpholine
1-methyl-1'-[3-(1-methylpiperidin-2-yl)propanoyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-(2-phenylethyl)-3-(1H-pyrazol-1-yl)-N-(pyridin-2-ylmethyl)benzamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pent-4-enamide
1-[1-(cyclopropylmethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
(2S)-2-acetamido-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-3-(1H-imidazol-4-yl)propanamide
ethyl 1-[(2-ethylphenyl)carbamoyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
2-[(4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}phenyl)formamido]acetamide
3-[(2H-1,3-benzodioxol-5-yl)amino]-N-(2-phenylethyl)piperidine-1-carboxamide
N-[(1-propyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-2-yl)acetamide
2-methyl-4-[4-(1-methyl-1H-1,2,4-triazol-5-yl)phenyl]butan-2-ol
N-[(5-fluoro-2-methylphenyl)methyl]-5-[4-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
N-(1-hydroxypropan-2-yl)-4-[(3-methoxypropyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
ethyl 1-({3-[(1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-3-yl)methoxy]phenyl}methyl)piperidine-4-carboxylate
5-{[4-(5-chloropyridin-2-yl)piperazin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine
N-[(6-hydroxypyrimidin-4-yl)methyl]-2-(1-propylpiperidin-4-yl)acetamide