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1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]but-3-en-1-one
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-4-(1H-1,2,3,4-tetrazol-1-yl)butanamide
3-{[1-(6-aminopyrimidin-4-yl)piperidin-4-yl]methyl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(1R,2S)-N1-butyl-N2-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]cyclohexane-1,2-dicarboxamide
1-[(2-ethylpyrimidin-5-yl)methyl]-N-[3-(4-fluorophenyl)phenyl]piperidine-3-carboxamide
5-(3-acetylphenoxymethyl)-N-methyl-N-(pyrimidin-4-ylmethyl)-1,2-oxazole-3-carboxamide
4-tert-butyl-N-{3-[4-(morpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}benzamide
{[3-(difluoromethoxy)phenyl]methyl}(methyl){[1-(propan-2-yl)piperidin-3-yl]methyl}amine
{3-[2-(2H-1,3-benzodioxol-5-yl)phenoxy]propyl}(methyl)amine
(3R,7S,8aS)-7-{[(3-fluorophenyl)methyl]amino}-3-[(1S)-1-hydroxyethyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
(3R,4R)-1-(1H-1,2,3-benzotriazole-5-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
4-{2-[1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-2-yl]ethyl}phenol
1-(carbamoylmethyl)-N-[(3-chloro-1-benzothiophen-2-yl)methyl]-N-methylpiperidine-4-carboxamide
4-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidin-2-amine
(4-{[(2-amino-5-ethyl-6-methylpyrimidin-4-yl)amino]methyl}phenyl)methanol
1-(3-{3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazol-5-yl}phenyl)ethan-1-one
2-(4-fluorophenoxy)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
2-ethyl-N-methyl-N-(quinoxalin-2-ylmethyl)pyrimidine-5-carboxamide
2-(1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}piperidin-3-yl)-1H-1,3-benzodiazole
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[(3S)-2-oxoazepan-3-yl]acetamide
N-ethyl-2-(pyridin-4-yl)benzamide
5-acetyl-N-methyl-N-[(5-phenyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-chlorobenzamide
2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-[2-(3-phenylpiperidin-1-yl)ethyl]acetamide
methyl (2R)-2-{[4-(4-methoxyphenoxy)phenyl]formamido}propanoate
(1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methanol
6-methyl-1-(3-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propyl)-1,2-dihydropyridin-2-one
3-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl}-N,N-dimethylaniline
4-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-3-(4-fluorophenyl)piperazin-2-one
3-(3-benzyl-1H-1,2,4-triazol-5-yl)-1-methyl-1-[(2-methylpyridin-4-yl)methyl]urea
3-methyl-1-[(4-methylphenyl)methyl]-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperazin-2-one
(2-methoxyethyl)({[4-phenyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl})(propan-2-yl)amine
5-{[3-(4-fluorophenyl)oxolan-3-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
propyl 2-({methyl[(3-methylthiophen-2-yl)methyl]amino}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxylate
5-(4-chlorophenyl)-N-{[4-(trifluoromethyl)phenyl]methyl}-1,2,4-triazin-3-amine
3-methyl-6-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)pyridazine
6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-{2-[4-(trifluoromethyl)phenyl]ethyl}piperidine-3-carboxamide
4-cyano-N-(3-ethoxy-2-hydroxypropyl)-1-methyl-1H-pyrrole-2-carboxamide
dimethyl(2-{[(3-methylthiophen-2-yl)methyl]({[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl})amino}ethyl)amine
4-(cyclohexylmethyl)-1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-1,4-diazepan-5-one
5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-2-(4H-1,2,4-triazol-4-yl)pyridine
3-chloro-N-cyclopentyl-4-{[1-(2-hydroxyacetyl)piperidin-4-yl]oxy}benzamide
4-{[1-(isoquinoline-1-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
2-{5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1H-pyrazole-3-carbonyl}-1,2,3,4-tetrahydroisoquinoline
2-{4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
5-(furan-3-ylmethyl)-3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)-2-(propan-2-yloxy)propanamide
methyl 1-[2-hydroxy-3-(3-{[(oxan-4-yl)amino]methyl}phenoxy)propyl]piperidine-4-carboxylate
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-oxo-2,3-dihydro-1,3-benzoxazole-6-sulfonamide