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2-(4-methylphenoxy)-N-{3-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}acetamide
2-methyl-6-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-one
5-oxo-1-{3-oxo-3-[4-(propan-2-yl)piperazin-1-yl]propyl}pyrrolidine-3-carboxylic acid
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)(2-methylpropyl)amine
3-{5-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazol-3-yl}pyridine
1-(4-{3-[(cyclooctylamino)methyl]pyridin-2-yl}piperazin-1-yl)ethan-1-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-(1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)propanamide
2-{8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-N-[2-(4-fluorophenyl)ethyl]acetamide
(4aR,7aS)-1-(2-methoxyethyl)-4-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(6-methoxynaphthalen-2-yl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}morpholine
4-{[4-(2-chlorophenyl)-4H-1,2,4-triazol-3-yl]methyl}pyridine
N,N,2-trimethyl-7-(4-methylpiperidine-4-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
4-methoxy-2-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenol
1-[2-methoxy-4-({methyl[(1-methylpiperidin-4-yl)methyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
7-(7-fluoro-4-methylquinolin-2-yl)-4-(furan-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-[2-(2-carboxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]pyrimidine-4-carboxylic acid
2-[(3-methoxyphenyl)amino]-N-(2-phenoxyethyl)butanamide
5-tert-butyl-3-[8-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]-1H-pyrazole
1-cycloheptyl-1H-1,2,3-triazole-4-carboxylic acid
4-(naphthalen-2-yloxy)-1-(oxan-4-yl)piperidine-4-carboxylic acid
5-({[4-methyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}methyl)-2-(trifluoromethyl)pyridine
(4aS,8aR)-6-(5-fluoropyrimidin-2-yl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[(5-methoxy-1H-indol-2-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
2-chloro-N-{2-[(3-ethyl-1,2-oxazol-5-yl)formamido]ethyl}benzamide
8-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
4-(benzyloxy)-1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
4-(morpholin-4-yl)-N-(2-phenylphenyl)piperidine-1-carboxamide
1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-4-(2-phenoxyethyl)piperazine
methyl(3-methylbut-2-en-1-yl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
1-[2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-4-methylpiperazine
2-methoxy-3-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
N-{2-[3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]propyl}-2-(trifluoromethyl)benzamide
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
1-[3-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propyl]piperidin-4-ol
3-{[(1-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperidin-4-yl)oxy]methyl}pyridine
2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}quinoxaline
5-chloro-2-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-(4-methyl-1H-imidazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[(quinolin-8-yloxy)methyl]-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1,3-oxazole-4-carboxamide
3-[(dimethylamino)methyl]-1-[(1-methyl-1H-indol-2-yl)methyl]piperidin-3-ol
methyl 5-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-{2-[3-(pyridin-2-yl)propanoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxolane-2-carboxamide
5-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-N,N-dimethylpyrimidin-2-amine
(4aR,8aR)-2-methanesulfonyl-7-[6-(methoxymethyl)pyridine-2-carbonyl]-decahydro-2,7-naphthyridin-4a-ol
N-[3-(4-methylpiperazin-1-yl)propyl]-4-(piperidin-3-yl)benzamide
2-chloro-5-acetamido-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}benzamide
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-methyl-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[7-(2H-1,3-benzodioxole-5-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1-phenylmethanesulfonamide
3-hydroxy-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}pyridine-2-carboxamide