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N-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
ethyl 1-(isoquinolin-5-ylmethyl)-4-(2-phenylethyl)piperidine-4-carboxylate
3-(1H-1,3-benzodiazol-1-yl)-N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)propanamide
N-[3-(4-ethoxyphenyl)propyl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide
3-[(3R,4S)-1-[(4-methylphenyl)carbamoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-[1-(propan-2-yl)piperidine-4-carbonyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
methyl(3-methylbutyl){[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
N-(1-{7-[(4-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
4-(2,1,3-benzothiadiazole-4-sulfonyl)-9-methoxy-7-[5-(trifluoromethyl)pyridin-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3R,4S)-4-cyclopropyl-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-amine
[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl](quinolin-5-ylmethyl)amine
N-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-6-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
4-[4-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperazin-1-yl]quinazoline
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(3-methylpyrazin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-phenoxy-1-{1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octan-6-yl}propan-1-one
4-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-phenylquinazoline
2-[({1-[(2-fluorophenyl)methyl]piperidin-3-yl}amino)methyl]phenol
[3-(2-methoxyethyl)-1-(5-propylthiophene-3-carbonyl)piperidin-3-yl]methanol
N-cyclopentyl-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-benzyl-N-(3-hydroxy-2-methylpropyl)acetamide
(benzylsulfamoyl)({[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl})amine
4-(5-ethylfuran-2-yl)-3-methyl-4H,5H,6H,7H-[1,2]thiazolo[5,4-b]pyridin-6-one
3-benzyl-4-[4-(1H-pyrazol-4-yl)butanoyl]piperazin-2-one
7-(3,5-dichloro-2-hydroxybenzenesulfonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[2-(3-fluoro-4-methylphenyl)pyrimidin-4-yl]pyrrolidin-3-ol
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-(1,2-oxazol-3-ylmethyl)-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
{[4-(furan-2-yl)phenyl]methyl}[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}[(dimethyl-1,2-oxazol-4-yl)methyl](2-methoxyethyl)amine
4-[(2-{1-[2-(prop-2-en-1-yloxy)benzoyl]piperidin-3-yl}-1H-imidazol-1-yl)methyl]pyridine
N-methyl-1-[2-(piperidin-1-yl)ethyl]-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}amine
(3S,7S)-5-[3-(ethylsulfanyl)propanoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
methyl 3-(2-chlorobenzamido)-6-[(4-methylpiperidin-1-yl)methyl]thieno[2,3-b]pyridine-2-carboxylate
3-[1-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-1-{[3-(trifluoromethoxy)phenyl]methyl}urea
N4-{imidazo[1,2-a]pyridin-3-ylmethyl}-N2,N2,5,6-tetramethylpyrimidine-2,4-diamine
1-methoxy-8-[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-(thiomorpholin-4-yl)acetic acid
5-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-[2-(pyridin-2-yl)ethyl]pentanamide
({5-[2-(4-chlorophenyl)morpholine-4-carbonyl]furan-2-yl}methyl)dimethylamine
5-methyl-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)pyridine-3-carboxamide
(4aS,8aR)-6-(1-benzofuran-2-sulfonyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
4-[4-(2-methoxyethoxy)phenyl]-N-methylbenzamide
5-{3-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
5,7-dimethyl-N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-cyclohexyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
2-(8-methylquinolin-5-yl)pyridine-4-carboxamide
1-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-4-(1H-pyrazol-3-yl)piperidine
1-[7,8-dimethyl-2-(pyrimidin-5-yl)quinoline-4-carbonyl]piperidine-3-carbonitrile
4-[1-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carbonyl]morpholine