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N-phenyl-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]({[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl})amine
(2R,3R,6R)-5-(1-benzofuran-3-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
(3S,4R)-4-(3-methoxyphenyl)-1-(quinoline-3-carbonyl)pyrrolidine-3-carboxylic acid
3-({4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzonitrile
1-methanesulfonyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]piperidin-4-amine
4-({methyl[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]amino}methyl)-1H-pyrrole-2-carbonitrile
N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
3-(4-chlorophenyl)-5-(oxan-4-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-(1-methylpiperidin-4-yl)-N-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-amine
4-{5-amino-4-cyano-1,6-diazatricyclo[6.2.2.02,7]dodeca-2(7),3,5-trien-3-yl}-N-methylbenzene-1-sulfonamide
{2-[3-(2-methylphenyl)piperidin-1-yl]-1,3-thiazol-4-yl}methanol
1-cyclopropyl-N-methyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-6-oxopiperidine-3-carboxamide
1-[4-(3,4-dichlorophenyl)piperazin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-4-sulfamoylbutanamide
3-{[(cyclopropylcarbamoyl)methyl]sulfamoyl}-N-(1-methoxypropan-2-yl)benzamide
1-{[3-(5-chloro-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
1-[2-(1H-imidazol-2-yl)benzoyl]-2-(3-methoxypropyl)piperidine
2-{4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-1,2,3-benzotriazole-5-carboxamide
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]acetamide
7-amino-4-(3-chloro-4,5-dimethoxyphenyl)-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
methyl 5-[(cyclohex-3-en-1-ylmethyl)amino]-3-acetamido-1-[2-(4-methoxyphenyl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[4-(5-ethyl-2-methylpyrimidin-4-yl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
N-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N-cyclopentyl-4-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}-4-oxobutanamide
2-(furan-2-yl)-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N,1-dimethyl-6-(2-phenylethyl)-N-(pyridin-3-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(1H-indol-5-ylmethyl)-decahydro-1,6-naphthyridin-2-one
7-(5-methylthiophen-2-yl)-9-(oxan-2-ylmethoxy)-4-propyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3S,9aR)-3-[(benzyloxy)methyl]-8-(4-phenylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
butyl 3,9-diazaspiro[5.6]dodecane-9-carboxylate
1-[1-(1H-pyrazole-3-carbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
{[4-(1H-imidazol-1-yl)phenyl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
N-cyclohexyl-1-{2-[(4-methoxyphenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methylpiperidine-3-carboxamide
N-(cyclopropylmethyl)-6-(4-methoxyphenyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(2S,4R)-N-(propan-2-yl)-4-(4-{[(pyrrolidine-1-sulfonyl)amino]methyl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxamide
N-cyclopentyl-4-(5-fluoropyridin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[2-(dimethylamino)butanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
6-methoxy-N4-methyl-N4-[(1-phenyl-1H-pyrazol-4-yl)methyl]pyrimidine-2,4-diamine
3-[2-(methylsulfanyl)benzoyl]-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidine
4-phenyl-1-[4-(pyrrolidin-1-ylmethyl)benzoyl]piperidin-4-ol
1-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)-4-[3-(trifluoromethyl)phenyl]piperazine
1-(2-phenylethyl)-N-[2-(1,3-thiazol-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-(3-chlorophenyl)-4-[1-(furan-3-carbonyl)piperidin-3-yl]piperazine
N-(2-oxo-2,3-dihydro-1H-indol-5-yl)benzamide
4-(1H-indol-2-ylmethyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-2-(3-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetamide
2-chloro-4-{[4-(hydroxymethyl)-4-(3-phenylpropyl)piperidin-1-yl]methyl}phenol
3-fluoro-N-{[(2S,4S)-4-fluoro-1-[2-(methylamino)acetyl]pyrrolidin-2-yl]methyl}benzene-1-sulfonamide