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N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-5-fluoro-N-methylquinazolin-4-amine
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-(4-methyl-3-phenylpiperazin-1-yl)ethan-1-one
2-(dimethyl-1,3-thiazol-5-yl)-1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]ethan-1-one
6-methyl-4-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
(2S)-1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(4,6-dimethylpyrimidin-2-yl)methyl]benzamide
(2S,4S)-4-[3-(2-amino-1,3-thiazol-4-yl)propanamido]-N,N-diethyl-1-methylpyrrolidine-2-carboxamide
N-[(5-methoxy-1H-indol-2-yl)methyl]-2-methyl-6-(piperidin-4-yl)pyrimidin-4-amine
3-{2-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
3,3-dimethyl-4-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperazin-2-one
6-methoxy-1-[(4-methoxyphenyl)methyl]-4-[3-(pyrazin-2-yl)propanoyl]-1,4-diazepan-2-one
N-({1-[ethyl(methyl)amino]cyclohexyl}methyl)-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
6-[(diethylamino)methyl]-N-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
ethyl 1-ethyl-5-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(1S,5R)-6-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
2-(dimethylamino)-N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-2-(3-methylphenyl)acetamide
7-[(4Z)-hept-4-en-1-yl]-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-{[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenol
2-[4-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)piperazin-1-yl]-N-ethylacetamide
N-[(2-methylphenyl)methyl]-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}acetamide
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carboxamide
(4aR,7aS)-N,N-dimethyl-4-(3-methyl-1H-pyrazole-5-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
(2-methylpropyl)[(3-phenyloxolan-3-yl)methyl](pyridin-2-ylmethyl)amine
8-(2-methoxy-5-methylbenzoyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-[(3-fluorophenyl)methyl]-3-(2-methoxyethyl)-5-{1-[2-(thiophen-2-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
4-{4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperazin-1-yl}-2-[2-(3-methoxyphenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
2-[2-(benzyloxy)phenyl]-1-(6-hydroxy-1,4-oxazepan-4-yl)ethan-1-one
(3R,9aR)-8-(2,5-dimethylbenzenesulfonyl)-3-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[(2-fluorophenyl)methyl]-3-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]piperazin-2-one
2-(piperidin-1-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
2-(4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-sulfonyl}phenoxy)acetamide
1-{3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
(5S,9aS,9bS)-5-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-{[(furan-3-ylmethyl)(methyl)amino]methyl}-N-(1-methyl-1H-1,2,3-triazol-4-yl)benzamide
[4-fluoro-7-(4-methoxy-2,5-dimethylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
5-methyl-N-(3-phenylpropyl)-6-(thiomorpholine-4-carbonyl)thieno[2,3-d]pyrimidin-4-amine
N-[3-(2-ethoxyphenyl)propyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
2-[(3R)-3-hydroxy-3-phenylpropyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
1-[(4-methoxyphenyl)methyl]-5-(pyridine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[(3S,5S)-5-(diethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]pyridine-3-carboxamide
4-[4-(1-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]piperidine
(1S,6R)-9-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-3,9-diazabicyclo[4.2.1]nonane
2-[(2-{[1-(2-methoxyphenyl)propan-2-yl](methyl)carbamoyl}phenyl)amino]acetic acid
3-{1-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]piperidin-4-yl}-1,3-oxazolidin-2-one
5-ethyl-N-methyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrimidin-2-amine
3-[3-(1H-imidazol-2-yl)benzoyl]-7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine
5-[({[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
1-[2-(piperazin-1-yl)ethyl]-N-(pyridin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide